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2-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-6-methylpyridine
2-methoxy-1-[1'-(1-methyl-1H-imidazole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-({2-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-4-methoxyphenyl}methyl)-1,4-diazepan-5-one
(2-{[4-(4-methylpyrimidin-2-yl)piperazin-1-yl]methyl}phenyl)methanol
1-[(2S)-2-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-1-yl]ethan-1-one
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(2-hydroxybutyl)propanamide
N-[(3R,4S)-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
5-cyclobutanecarbonyl-1'-(pyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(2-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-oxoethyl)-1,2,3,4-tetrahydroquinolin-2-one
2-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-7-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinoline
4-methyl-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}piperidine-4-carboxamide
3-chloro-4-{[4-(2,5-dimethylpyrimidin-4-yl)piperazin-1-yl]methyl}phenol
7-(1-benzothiophen-3-yl)-4-[(2-methylpyrimidin-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(5-{imidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl)-1H-pyrazole
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazole
3-{[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}propane-1,2-diol
1-[4-(3-chloropyridin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
6-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]pyridine-2-carbonitrile
4-[5-(3-phenylpropanamido)-1H-pyrazol-1-yl]-N-(prop-2-en-1-yl)piperidine-1-carboxamide
(3R,4R)-1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
2-(cyclopent-2-en-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]ethan-1-one
(9aS)-N-[3-(benzyloxy)phenyl]-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxamide
N-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(1,2,3,6-tetrahydropyridin-4-yl)ethan-1-one
3-(propan-2-yl)-4-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]piperazin-2-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(cyclopropylmethyl)acetamide
N,5,6-trimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]pyridine-3-carboxamide
N-{1-[1-(3-methylbut-2-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
(3S,7S)-5-[3-(dimethylamino)benzoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-[(cyclohexylmethyl)amino]-N-methylpyrrolidine-2-carboxamide
N-(dimethyl-1,2-oxazol-4-yl)-3-{[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzamide
1-(4-{[(1,3-benzoxazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
2-methyl-N-(2-{7-[2-(4-methylphenoxy)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
[(2,2-dimethyloxan-4-yl)methyl]({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
2-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]-1-methyl-1H-1,3-benzodiazole
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)pyrazolo[1,5-a]pyridine-3-carboxamide
5-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-4-ethyl-1,2,3-thiadiazole
2-(2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
5-(2,5-dimethylphenoxymethyl)-N-[(3-methoxyphenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-(cycloheptylamino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2,6-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
3-(azepane-1-carbonyl)-1-ethyl-N-(2-methoxyethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(1S,5R)-6-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-[2-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-3-phenylcyclopent-2-en-1-one
2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-(3-phenylpropyl)acetamide
methyl (2S,4R)-1-[(2,4-dimethylphenyl)methyl]-4-(3-methoxybenzamido)pyrrolidine-2-carboxylate
3-(1H-1,3-benzodiazol-2-yl)-N-[1-(2-methylpropyl)-1H-pyrazol-5-yl]azetidine-1-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-(1-benzothiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one