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N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
5-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
1-({2-[3-(piperidin-1-yl)propoxy]phenyl}methyl)piperidin-3-amine
8-methyl-4-(4-methyl-1,4-diazepane-1-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-[2-(dimethylamino)ethyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-[(3-methoxyphenyl)methyl]-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
(3R,4S)-4-cyclopropyl-1-(quinoline-6-carbonyl)pyrrolidin-3-amine
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2-methoxyphenyl)ethan-1-one
(4-{[2-(5-methylfuran-2-yl)phenyl]methyl}morpholin-3-yl)methanol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
(2,1,3-benzoxadiazol-5-ylmethyl)({[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(pyridin-2-yl)pyrimidine
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
6-[3-(3-methylphenyl)benzoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-ethyl-5-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyrimidin-2-amine
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
4-{[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-N-methylbenzamide
6-methoxy-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-ethyl-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(carbamoylmethyl)-N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
1-[3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzenesulfonyl]-1,4-diazepan-5-one
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-hydroxy-2-(4-methylphenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}pyrimidine-5-carboxamide
8-[(2,6-dichloro-3-hydroxyphenyl)methyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
2-(4-fluorophenyl)-4-[5-(propan-2-yl)pyrimidin-4-yl]morpholine
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}-1-(propan-2-yl)piperidine-4-carboxamide
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
{4-[(3-chloro-4-methoxyphenyl)methyl]morpholin-3-yl}methanol
3-(3-acetylphenyl)-1-methyl-6-(1,2,5-thiadiazole-3-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-{[3-({2-[(3-methylpyridin-2-yl)amino]ethyl}carbamoyl)phenyl]amino}acetic acid
{1-[5-(cyclopentylamino)-5,6,7,8-tetrahydroquinazolin-2-yl]piperidin-4-yl}methanol
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
ethyl[(2-fluorophenyl)methyl][(4-methyl-1H-imidazol-5-yl)methyl]amine
methyl 3-[(quinolin-6-ylformamido)methyl]-5-[2-(thiophen-3-yl)acetamido]benzoate
1-[4-(4-aminoquinazolin-6-yl)phenyl]-3-ethylurea
(2R,3R)-3-[4-(2-hydroxyphenyl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(1H-imidazol-2-ylmethyl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1,4-diazepan-6-ol
(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}morpholin-2-yl)methanamine
(2S)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-4-methylpentanamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1-phenylmethanesulfonamide
N-(dimethyl-1,2-oxazol-4-yl)-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholine-4-carboxamide
1'-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]