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N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
3-(3-fluorophenyl)-1-methyl-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
1-{2-[({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-pyrrol-1-yl)propan-1-one
7-methoxy-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)piperidin-4-ol
2-[4-(3-cyclopentylpropyl)piperazin-1-yl]-6-(pyrrolidine-1-carbonyl)pyrazine
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-benzyl-2-(3,3-dioxo-1,3λ6,4-oxathiazinan-4-yl)acetamide
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-[1-(2-methylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
(1R,3S)-7-[(4-fluoro-3-methoxyphenyl)methyl]-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}acetic acid
(3aS,6aR)-5-[(5-ethylpyridin-2-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(2,6-difluorophenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[4-(ethylamino)pyrimidin-2-yl]piperidine-4-carboxamide
6-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-ylmethyl]-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
4-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-1-(4-fluorophenyl)butan-1-one
4-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
(4aS,8aR)-6-(2-methoxyacetyl)-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-[2-(2-chloro-4-methylphenoxy)ethyl]pyrimidine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]ethan-1-one
2-(2-hydroxyethyl)-8-[(2,4,6-trifluorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}quinolin-8-ol
5-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazole
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-6-methylpyridine-3-carbonitrile
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(thiophen-3-yl)propanamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-hydroxypyridine-3-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
4-(azonan-1-yl)-N-[2-(diethylamino)ethyl]pyridine-2-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2,3,5-trimethyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-{[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]sulfonyl}-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
3-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
2-methoxy-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
2-[4-(2-ethoxypyridine-3-carbonyl)morpholin-3-yl]-N-(2-fluorophenyl)acetamide
4-[4-(1H-1,3-benzodiazol-2-yl)-1H-1,2,3-triazol-1-yl]-1-propylpyrrolidin-2-one
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
2,6,8-trimethyl-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]quinoline
5-methanesulfonyl-N,2-dimethyl-N-[(5-methylthiophen-2-yl)methyl]pyrimidin-4-amine
2-(4-chlorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-methyl-N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}pyridazin-3-amine
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(3-hydroxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-2-methyl-1,3-thiazole
3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-one
1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
(1S,5R)-6-(2-methoxyethyl)-3-[3-(1H-pyrazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one