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2-[5-(1-acetamido-2-methylpropyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]benzoic acid
N-cyclopropyl-7-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-(furan-2-yl)-N-(oxolan-2-ylmethyl)propanamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-(4-ethoxy-3-methylphenyl)-4-[4-(1H-imidazol-2-yl)piperidin-1-yl]butane-1,4-dione
4-phenyl-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]azepane
(3R,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
5-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
1-(2-methoxyphenyl)-4-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-one
2-[4-(dimethylamino)butyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[1-(4-chlorophenyl)cyclobutanecarbonyl]-9-(oxan-2-ylmethoxy)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{2-[1-(4-tert-butylbenzoyl)piperidin-2-yl]ethyl}-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
N-{[3-(butan-2-yloxy)phenyl]methyl}-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-[4-(pyridin-3-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-pyrrole-2-carboxamide
(5S,9aS,9bS)-5-(furan-2-yl)-2-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl 2-{methyl[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]carbamoyl}piperidine-1-carboxylate
1-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-amine
1-(cyclohexyloxy)-3-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)propan-2-ol
1-cyclohexyl-4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperazin-2-one
1,3-dimethyl-5-{2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)oxane-4-carboxamide
(2S,4S)-N-ethyl-1-(furan-2-ylmethyl)-4-(3-methoxypropanamido)pyrrolidine-2-carboxamide
1-benzyl-N3-cyclopropyl-N5-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3S,4R)-1-(4-chloro-2-methoxybenzoyl)-4-propylpyrrolidin-3-yl]acetamide
(1R,5R)-6-(2-methoxyethyl)-3-(2-methyl-5-propylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
4-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridin-2-amine
4-(2,4-difluorophenyl)-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{3-[2-amino-3-cyano-6-(1H-pyrrol-2-yl)pyridin-4-yl]-2-methyl-1H-indol-1-yl}acetamide
2-methyl-4-[(3,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(cyclopropylmethyl)-9-(1-ethyl-1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-4-cyclopropyl-1-(dimethylcarbamoyl)pyrrolidin-3-yl]-5-methoxy-1H-indole-2-carboxamide
methyl 4-({[(3S,5S)-1-[(4-chlorophenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidin-3-yl]amino}methyl)benzoate
4-methoxy-2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenol
3-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-N-(1,3-thiazol-2-yl)propanamide
3-(propan-2-yl)-5-{1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-2-yl}-1,2,4-oxadiazole
N3-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N1-(5-methylpyridin-2-yl)propane-1,3-diamine
1-(2-{methyl[3-(5-methylfuran-2-yl)butyl]amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[2-(2-methoxypyridin-3-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
N-(3-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-3-oxopropyl)-N-methylmethanesulfonamide
2-(1-{[1-(5-fluoro-2-methylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
1-(4-{[4-(2,6-dimethylquinoline-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
5-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
3-({1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
1-[(2-chloro-6-fluorophenyl)methyl]-5-(1,4-dioxan-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
2-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-5-methoxy-4H-pyran-4-one
5-[1-ethyl-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]-1-(2-methoxyethyl)piperidin-2-one
3-{2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
1-(3-chloro-4-ethoxyphenyl)-3-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}urea
4-[(E)-2-(furan-2-yl)ethenyl]-3-methyl-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one