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(3-{2-[1-(furan-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-methyl-8-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(3R,4R)-1-(2-methyl-1,3-benzothiazole-6-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]quinoline
methyl({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl})[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
1-methyl-3-(pyrrolidine-1-carbonyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-phenylbenzamide
3,3-dimethyl-1-({5-[(3-methyl-1H-indol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
1-methyl-2-[1-(1,3-thiazol-4-ylmethyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
1-[(2-fluorophenyl)methyl]-N-(pyridin-2-ylmethyl)piperidin-3-amine
2-(4-propanoylphenoxy)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-(cyclopropylmethyl)-3-{[4-(ethanesulfonyl)piperazin-1-yl]methyl}-3-hydroxypiperidin-2-one
N-methyl-2-(3-methyl-3-phenylpiperidin-1-yl)-N-phenylacetamide
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
2-(butylsulfanyl)-N4-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}pyrimidine-4,6-diamine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[(3R,4S)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[(4-fluorophenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[(3R,4S)-1-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
6-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-{[1-(pyridine-3-sulfonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
7-(oxan-4-yl)-2-(1H-1,2,3-triazol-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
[(2-ethyl-3-methyl-1H-indol-5-yl)methyl][(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amine
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1-(propan-2-yl)piperidine-4-carboxamide
4-[(4-ethoxyphenyl)methyl]-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
7-(2-methoxyethyl)-2-(pyrimidin-2-yl)-2,7-diazaspiro[4.5]decane
N-(1,2-oxazol-3-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[1'-(1-ethylpiperidine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-[2-(morpholin-4-yl)ethyl]-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)piperidin-2-one
3-(cyclopropylmethyl)-1-(4-oxo-4-phenylbutanoyl)piperidine-3-carboxylic acid
1-cyclopentyl-4-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]pyrrolidin-2-one
[1-(4-fluorobenzoyl)-3-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
(1-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-2,5-dihydro-1H-pyrrol-2-yl)methanol
1-(4-benzylpiperazin-1-yl)-3-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]propan-1-one
5-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]azepan-2-one
5-amino-4-chloro-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1H-pyrazole-3-carboxamide
5-fluoro-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyrimidin-4-ol
methyl 6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-3-(thiophene-3-amido)thieno[2,3-b]pyridine-2-carboxylate
6-methyl-2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}quinolin-4-ol
2-(4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
ethyl 4-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}piperazine-1-carboxylate
3-(3-fluorophenyl)-4-(2-phenylpyrrolidine-1-carbonyl)-1H-pyrazole
(3S,4S)-4-cyclopropyl-1-{[6-(dimethylamino)pyridin-3-yl]methyl}pyrrolidine-3-carboxylic acid