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5-methyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
(1R,6S)-3-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
1-(piperidin-3-ylmethyl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[3-(pyrrolidin-1-yl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
{2-ethoxy-5-[(4-ethoxypiperidin-1-yl)methyl]phenyl}methanol
N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(7-methyl-3-{[(2-phenylethyl)amino]methyl}quinolin-2-yl)piperidin-4-ol
2-[(4aR,7aS)-4-[(2-methylpyrimidin-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
N-(2-methanesulfonylethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-methyl-N,N-bis(prop-2-en-1-yl)-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
(3S,4R)-1-(1,4-dithiepan-6-yl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-4-[(dimethylamino)methyl]piperidin-4-ol
N,2-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(thiophen-2-ylformamido)propanamide
3-{[(3-methyl-1H-pyrazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}propan-1-ol
1-[3-(3-fluorophenyl)phenyl]-N-[2-(pyrazin-2-yl)ethyl]piperidin-4-amine
2-(dimethylamino)-N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)benzamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-one
1-methyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-dihydropyridin-2-one
(2S,4S,5R)-1,2-dimethyl-4-{methyl[(3-methylpyridin-2-yl)methyl]carbamoyl}-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
1-{5-[(4-ethyl-1,4-diazepan-1-yl)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
(2S)-2-acetamido-N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-(2-methylphenyl)-1-(1,2-oxazolidin-2-yl)-3-phenylpropan-1-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(pyrrolidin-1-yl)piperidine
N,3,6,7-tetramethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1-benzofuran-2-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
methyl 1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
(2S,4R)-4-(2,5-dimethylfuran-3-amido)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
N-(2-chlorophenyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
2-(4-methyl-6-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]amino}pyrimidin-2-yl)phenol
N-(2-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methylbenzamide
ethyl 2-{[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]amino}acetate
(2S,4R)-4-amino-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-oxo-4-phenylbutanamide
4-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-(2-methoxyethyl)pyrrolidin-2-one
1-(4-{[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]methyl}phenyl)pyrrolidin-2-one
N-(1-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
4-methyl-2-{2-oxo-2-[4-(pyridin-4-yl)piperazin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
1-(2-methoxyacetyl)-N-methyl-N-(quinolin-2-ylmethyl)piperidine-4-carboxamide
2-(cyclohex-1-en-1-yl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
N-[2-(2-chlorophenyl)-1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
6-chloro-3-[5-chloro-2-(propan-2-yloxy)phenyl]-[1,2,4]triazolo[4,3-a]pyridine
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-3-(1H-pyrazol-1-yl)benzamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-(2-fluorophenyl)cyclopropane-1-carboxamide
3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-4-[(2-methylphenyl)methyl]piperazin-2-one