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N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-oxobutanamide
4-({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)piperazin-2-one
({4-[(dimethylamino)methyl]phenyl}methyl)(1H-imidazol-4-ylmethyl)methylamine
2-[3-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)phenoxy]ethan-1-ol
2-(3-fluorophenyl)-8-methoxy-5-[(4-methyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
N,7,8-trimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)quinoline-4-carboxamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-amine
3-(3,4-dimethoxyphenyl)-N-{[5-fluoro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-(3,5-dimethylfuran-2-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
N-[3-(azepane-1-carbonyl)phenyl]-3-(pyridin-2-yl)azetidine-1-carboxamide
5-[3-(2-methoxyphenoxy)propyl]pyridine-3-carboxamide
6-(1-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-3-yl)pyrimidin-4-ol
(2S,4R)-4-(dimethylamino)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylic acid
methyl 4-[(8-methylquinolin-5-yl)carbamoyl]piperazine-1-carboxylate
N-{[4-(dimethylamino)oxan-4-yl]methyl}-3-(2-fluorophenyl)-3-phenylpropanamide
3-({[2-(dimethylamino)ethyl][(3-methylthiophen-2-yl)methyl]amino}methyl)-5-methyl-1H-indole-2-carboxylic acid
5-acetyl-3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-(4-fluorophenyl)butanamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(2-oxopiperidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
6-methyl-4-{4-[1-(piperidin-1-yl)ethyl]phenyl}-2,3-dihydropyridazin-3-one
2-methoxy-3-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
6-butyl-2-(4-{[(2,3-dihydroxypropyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-(methylsulfanyl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1,3-thiazole-4-carboxamide
(3S,5R)-N3-[(1-ethylpyrrolidin-2-yl)methyl]-N5-(4-fluorophenyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
3-{[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl][(4-chlorophenyl)methyl]amino}propan-1-ol
2-[(3-methoxyphenyl)amino]-N-[(5-methylpyrazin-2-yl)methyl]butanamide
3-[2-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethyl]phenol
7-chloro-3-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]quinolin-4-ol
5-[3-(methoxymethyl)-1H-1,2,4-triazol-5-yl]-2-methylquinoline
N6-(2-methoxyethyl)-N5-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methoxyethyl)piperidine
6-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[1-(thiophen-2-yl)propan-2-yl]propanamide
1-(4-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-phenyl-1,2-oxazole-4-carboxamide
2-{[9-(2-hydroxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]methyl}benzonitrile
1-{2-[1-(2-methylpyridin-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[3-(4-fluorophenyl)propyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
N-[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]-4-(1H-pyrazol-4-yl)butanamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]benzamide
2-({3-[3-(diethylcarbamoyl)piperidine-1-carbonyl]phenyl}amino)acetic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]piperidine-3-carboxamide
1-methyl-9-(prop-2-en-1-yl)-4-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-ethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]imidazo[1,2-a]pyridine-3-carboxamide
3-(2-methylphenyl)-1-(quinolin-2-ylmethyl)pyrrolidin-3-ol
2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-N,N-dimethylethane-1-sulfonamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(thiophene-2-carbonyl)piperidine