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6-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
N-{3-[({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)carbamoyl)methoxy]phenyl}propanamide
N-ethyl-3,5-dimethyl-1-(prop-2-en-1-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
4-{5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]furan-2-carbonyl}morpholine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1,5-trimethyl-1H-pyrazole-3-carboxamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-(1-methoxypropan-2-yl)piperidine-4-carboxylate
(2S,4R)-N-methyl-4-(4-{4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
5-{5-[2-(4-fluorophenyl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-2-(pyrazin-2-yl)ethan-1-one
(1S,5R)-6-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[(dimethylamino)methyl]-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-ol
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-(4-propanoylphenoxy)acetamide
1-(4-methoxybenzoyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazine
1-amino-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropane-1-carboxamide
3-(4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperazin-1-yl)propan-1-ol
methyl (2S,4R)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(dimethylamino)pyrrolidine-2-carboxylate
N-(1,3-dihydroxypropan-2-yl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-[3-(4-methylpiperazin-1-yl)butyl]pyrimidin-4-amine
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(1H-1,2,4-triazol-3-yl)benzamide
N-(4-butylphenyl)-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
1-{1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}-4-methyl-1,4-diazepane
3-[(3R,4S)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-(methylamino)-N-[1-(thian-4-yl)piperidin-4-yl]pyridine-4-carboxamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]piperidine
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(pyridin-3-yloxy)propyl]acetamide
N-({2-[2-(2,5-dimethylfuran-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2,3-dihydro-1,4-benzodioxine-2-carboxamide
(3R,4R)-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
methyl 4-oxo-4-[3-(4-phenoxybenzoyl)piperidin-1-yl]butanoate
4-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
4,7-dimethyl-2-[4-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]quinazoline
4-ethoxy-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)propanamide
6-methyl-1-{2-[3-(propan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydropyridin-2-one
(3S,4R)-1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{1-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]cyclohexyl}morpholine
{[5-(2H-1,3-benzodioxol-5-yl)-2-methoxyphenyl]methyl}(methyl)amine
3-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-N-cyclooctylacetamide
N-[2-(pyridin-2-yl)ethyl]-6-{2-[3-(trifluoromethyl)phenyl]acetyl}-6-azaspiro[2.5]octane-1-carboxamide
2,7-dimethyl-4-[3-(prop-2-en-1-yloxy)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2-{[(3,5-dichloropyridin-4-yl)methyl](methyl)amino}ethyl)piperidin-2-one
(2R,6R)-4-(3-acetamidopropanoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-5-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)pyridin-2-amine
[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl](ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
1-cyclobutanecarbonyl-4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidine
6-[(4-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-1H-1,2,3-triazol-1-yl)methyl]pyrimidin-4-ol
4-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)morpholine
1-(2-benzylphenyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole