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3-[2-(quinoxalin-5-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]phenol
1-(4-methyl-1,3-thiazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[(2-methoxyphenyl)methyl]benzamide
2-{1-benzyl-4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-2-methyl-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazine-1,1-dione
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(1,3-thiazol-2-yl)pyrrolidin-3-yl]methanol
2-(3-chloro-4-fluorophenoxy)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]ethan-1-one
1-ethyl-N,5-bis[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-cyclopropyl-3-{1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]piperidin-4-yl}propanamide
2-(1-methyl-1H-pyrazol-3-yl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine
6-oxo-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,6-dihydropyridine-2-carboxamide
5-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-ethoxy-1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}propan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
[1-methanesulfonyl-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
2-(2H-1,3-benzodioxol-5-yl)-2-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}acetic acid
3-[(3R,4S)-1-[3-(difluoromethoxy)benzoyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-{4-[({[2-(dimethylamino)pyridin-3-yl]methyl}amino)methyl]phenyl}acetamide
1-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)ethan-1-one
(3aS,6aS)-2-cyclopentyl-5-[2-(2-fluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2r,4r)-N-methyl-6,8-dioxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-5,7-diazaspiro[3.4]octane-2-carboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-phenylethyl)piperidine
(1-{[methyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl})amino]methyl}cyclopentyl)methanol
(1R,5S)-6-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-6-azabicyclo[3.2.1]octane
4-[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-(4-fluorophenyl)piperidin-4-ol
2-(4-{[2-(benzyloxy)phenyl]methyl}piperazin-1-yl)pyrimidine
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopentyl-1-(2-ethoxyethyl)-N-ethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-(3-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-oxopropyl)piperidin-2-one
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(3-methoxyphenoxymethyl)piperidine
3-[2-(2-hydroxyethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-(2-methoxyethyl)-1-[(2-methylphenyl)methyl]pyrrolidine-2-carboxamide
{1-[6-(aminomethyl)-2-methylpyrimidin-4-yl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
[(3R,4R)-1-[(3,4-difluorophenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-ethyl-2-(isoquinolin-5-yl)benzamide
N-(2-ethyl-1,3-dihydroxypropan-2-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1S,5R)-3-(2,4-dichlorobenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-1-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}piperidine-3-carboxamide
N-({7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
2-(1-{[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
N-(2-phenylethyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
3-[(dimethylamino)methyl]-1-(3,6-dimethylpyrazin-2-yl)piperidin-3-ol
(3aR,6aR)-2-methanesulfonyl-5-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-amino-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]pyridine-3-carboxamide
N-cyclopropyl-3-{5-[(3-methylthiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-chloro-N-{[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}pyridine-4-carboxamide