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1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-5-[2-(thiophen-2-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-(furan-2-ylmethyl)-N-methylacetamide
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]methyl}amine
1-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-4-amine
N-[2-(phenylsulfanyl)ethyl]-N-(propan-2-yl)-4-(1H-1,2,4-triazol-1-yl)butanamide
N-(2-hydroxyethyl)-4-[methyl({[3-(trifluoromethyl)phenyl]methyl})amino]pyridine-2-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-(2-oxopyrrolidin-1-yl)butanamide
N-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-1-(morpholin-4-yl)propan-1-one
[4-(2-ethylphenyl)pyridin-2-yl]methanol
N-[3-({[(2S)-2-hydroxy-2-phenylethyl]carbamoyl}amino)-2-methylphenyl]cyclopentanecarboxamide
5-methyl-3-{3-oxo-3-[4-(pyridin-4-yl)piperidin-1-yl]propyl}-2,3-dihydro-1,3-benzoxazol-2-one
(5-{1-[3-(1,3-benzothiazol-2-yl)propyl]-1H-imidazol-2-yl}furan-2-yl)methanol
(1H-imidazol-4-ylmethyl)(2-methoxyethyl)[(4-methylphenyl)methyl]amine
1-[1'-(2-propyl-1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
4-(methoxymethyl)-1-{[(1R,2R)-2-phenylcyclopropyl]methyl}piperidine
2-(1H-imidazol-2-yl)-N-[1-(thian-4-yl)piperidin-4-yl]benzamide
1-cyclopentyl-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]piperidine-3-carboxamide
1-[2-(dimethylamino)ethyl]-5-(5-methylpyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-({4-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)morpholine
2-[3-(dimethylamino)propyl]-9-[(2R)-2-hydroxy-2-phenylacetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 2-[4-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetate
6-chloro-N-cyclopentyl-2-(pyrimidin-5-yl)quinoline-4-carboxamide
(1S,5R)-3-{[6-(dimethylamino)pyridin-3-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-2-[methyl(phenyl)amino]-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-{[3-(4-benzoylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-2-methylpyridine
(3R,4R)-1-(2-cyclopropylpyrimidine-5-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-cyclopropyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-2-cyclopropyl-3,4-dihydropyrimidin-4-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
2-{[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]methyl}quinolin-4-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-(3-phenylpiperidin-1-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
[(3R,5R)-1-(6-cyclopropylpyrimidin-4-yl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
4-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]pyrimidine-5-carboxylic acid
3-{[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]methyl}-2-methoxy-4,6-dimethylpyridine
(3aR,6aR)-2-[(4-methylpiperidin-1-yl)sulfonyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(5-methylthiophen-2-yl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
N-(3-methoxypropyl)-1-methyl-5-(2,5,7-trimethylquinoline-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{3-[2-(azepan-1-ylmethyl)-4-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
N-[2-hydroxy-2-(3-phenoxyphenyl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(4-methoxyphenoxymethyl)-N-methyl-N-propyl-1,3-oxazole-4-carboxamide
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{2-[(3-fluorophenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-cyclobutyl-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-5-(2-methoxyacetamido)-N,1-dimethyl-1H-1,3-benzodiazole-7-carboxamide
8-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-[2-(dimethylamino)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1,3-thiazol-4-yl)ethyl]amine