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N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-5-[(methylsulfanyl)methyl]furan-2-carboxamide
3-chloro-6-[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyridine-2-carboxylic acid
9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-3-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-[1-(2-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
2-({[(3R,4R)-1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-[2-amino-3-cyano-6-(3,5-difluorophenyl)pyridin-4-yl]benzamide
(3S,4S)-4-methyl-1-(6-methylpyridazin-3-yl)piperidine-3,4-diol
2-{4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
(2E)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(pyridin-2-yl)prop-2-en-1-one
2-hydroxy-N-methyl-N-[(4-phenoxyphenyl)methyl]acetamide
5-[(2-chlorophenyl)methyl]-5-(1-cyclohexanecarbonylpiperidin-4-yl)-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-{2-[1-(2-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(2S)-2-amino-1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
N-[(3S,4R)-1-(2-oxo-4-phenylbutanoyl)-4-propylpyrrolidin-3-yl]acetamide
N-(butan-2-yl)-3,5-diacetamido-N-[(2-fluorophenyl)methyl]benzamide
methyl({[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
(3R)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-benzyl-5-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methylphenyl)methyl]piperidine
N-ethyl-5-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-amine
N-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(oxolan-3-yl)piperidine-4-carboxamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(oxan-4-yl)benzamide
{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-methyl-N-(quinolin-5-ylmethyl)propanamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}piperidin-2-one
1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(methylsulfanyl)pyridine-3-carboxamide
N-[(2S)-oxolan-2-ylmethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]-2-(2-methoxyethyl)morpholine
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
(1-benzofuran-2-ylmethyl)(ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
2-(2-{1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-(1-{7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
6-methoxy-3-methyl-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]-1-benzofuran-2-carboxamide
N-(2,5-dimethoxyphenyl)-2-propylpyrrolidine-1-carboxamide
2-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}ethoxy)ethan-1-ol
4-ethyl-3-[1-(4-methanesulfonylbenzoyl)piperidin-4-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(3-hydroxypiperidin-1-yl)ethyl]benzamide
3-({[2-(1-hydroxycyclopentyl)ethyl](methyl)carbamoyl}amino)-2-methyl-N-(2-methylpropyl)benzamide
4-ethyl-1-methyl-3-(1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-3-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
5-(3,4-dimethylphenoxymethyl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1,2-oxazole-3-carboxamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1H-imidazole-2-carboxamide
1-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
N-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
3-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione