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({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)bis(pyridin-3-ylmethyl)amine
{3-[(4-fluorophenyl)methyl]-1-[4-(methylamino)pyrimidin-2-yl]piperidin-3-yl}methanol
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(1-ethylcyclopropyl)methyl]-1H-pyrazole-3-carboxamide
5-[5-(2-ethylpyrimidin-5-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
N-[2-(3-fluorophenyl)ethyl]-7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(3-methoxypropyl)piperazine
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-(2-methanesulfonylethyl)piperidin-4-amine
3,5-dimethyl-1-{1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-3-yl}-1H-pyrazole
2,8-dimethyl-4-(3-methyl-1H-1,2,4-triazol-5-yl)quinoline
N-[(3R,4S)-4-cyclopropyl-1-(1-phenylpiperidin-4-yl)pyrrolidin-3-yl]-2-methoxyacetamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
6-methyl-2-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
N-[3-(1H-indazol-1-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1-{[methyl({[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}cyclopropyl)methanol
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
4-{methyl[(1-methylpiperidin-2-yl)methyl]carbamoyl}pyridin-1-ium-1-olate
N-[2-(2-chlorophenyl)ethyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
(1S,5R)-6-(2-methoxyethyl)-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-[6-(dimethylamino)pyridin-3-yl]-5-(morpholine-4-sulfonyl)benzoic acid
4-methyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]pyrimidin-2-amine
N-[2-(cyclohexylsulfanyl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-benzyl-3-{[1-(1,3-thiazol-2-yl)piperidin-4-yl]oxy}benzamide
3-({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)butan-1-ol
9-(morpholine-2-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
9-methoxy-4-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-{7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(1-methoxypropan-2-yl)pyridin-2-amine
3-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1-[3-(pyridin-3-yl)propyl]urea
N5-cyclopropyl-N6-[2-(pyridin-3-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-(4-benzyl-1H-pyrazol-5-yl)-1-(dimethyl-1,3-oxazole-5-carbonyl)piperidine
2-[({1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]-N-methylacetamide
N-{1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-4-yl}methanesulfonamide
3-chloro-N-cyclopentyl-4-{[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}benzamide
5-(4-fluorophenyl)-N-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-triazin-3-amine
N-[(3,5-dichloropyridin-4-yl)methyl]-N-methylthian-4-amine
N-ethyl-5-[2-(3-fluorophenyl)azepane-1-carbonyl]pyrimidin-2-amine
6-[3-(naphthalene-2-carbonyl)piperidin-1-yl]pyrazine-2-carboxamide
1-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-cyclopentylethan-1-one
1-[(diethylcarbamoyl)methyl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(pyrimidin-2-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
1-(2,4-difluorophenyl)-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-1H-1,2,4-triazole
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
1-[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,6-dimethylquinoline-4-carboxamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methoxypyridine-3-carboxamide
7-cyclohexyl-2-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-[1-(thiophen-2-yl)propan-2-yl]propanamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
4-{1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]azetidin-3-yl}pyridine