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1-{3-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-3-oxopropyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
8-[(3-phenylphenyl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
ethyl 1-(2,4-dimethylbenzoyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
N-(2,5-dimethylphenyl)-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
1-(2-{[2-(thiophen-2-yl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol
1-[(4aS,8aR)-4a-(hydroxymethyl)-6-propyl-decahydro-1,6-naphthyridin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
N-cyclohexyl-3-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]propanamide
1-(oxolan-2-ylmethyl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(4-fluorophenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-{4-[(4-ethynylphenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(3S,4R)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(4-methyl-1,3-thiazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
N-benzyl{[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]amino}sulfonamide
methyl 2-{[(2-chlorophenyl)methyl]sulfamoyl}-6-[2-(methylsulfanyl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[3-(2-methyl-1H-imidazol-1-yl)propyl]amine
3-(propoxymethyl)-N-[4-(pyridin-3-yloxy)phenyl]pyrrolidine-1-carboxamide
2-ethoxy-1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
3-(pyridin-4-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]propan-1-one
3-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-5-(2-methylphenyl)-1,2,4-triazine
ethyl 1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazole-2-carboxylate
3-benzyl-5-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole
1-(2-methoxyethyl)-4-phenyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
N-(2-methoxyethyl)-N-methyl-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
3-(4-benzylpiperazine-1-carbonyl)-2,8-diazaspiro[4.5]decane
3-[(2-methoxypyridin-3-yl)formamido]-N-(3-methylphenyl)propanamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
1-(4-{[(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amino]methyl}thiophen-2-yl)ethan-1-one
N-[2-(3-methoxyphenyl)-1-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-4-yl}ethyl]-N-methylpyridine-2-carboxamide
1-[(2-chlorophenyl)methyl]-N-[(3-methylpyridin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-4-carboxamide
1-[(4-chlorophenyl)methyl]-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]piperidin-2-one
N-benzyl-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-[(3-methylphenyl)methyl]piperidine-3-carboxylic acid
4-hydroxy-3-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
2-({[(3R,4R)-1-(3-chloro-4-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-(3-methoxypyrazin-2-yl)-5-methyl-1H-indole
N-[(3,4-difluorophenyl)methyl]-3-[1-(isoquinolin-5-ylmethyl)piperidin-3-yl]propanamide
methyl 1-[(3S,5S)-1-(furan-3-ylmethyl)-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N,N-dimethyl-2-[2-(2-methylpropyl)pyrimidin-5-yl]quinoline-4-carboxamide
2-[(4-chlorophenyl)methyl]-5-[3-(methoxymethyl)piperidine-1-carbonyl]-1,3-benzoxazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-6-(3-phenylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
(5S)-5-[({[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
5-(5-phenyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
{1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-3-ethylpiperidin-3-yl}methanol
N-{2-[4-(2,2-dimethylpropyl)morpholin-2-yl]ethyl}pyridine-4-carboxamide
N-(2-{7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide