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6-chloro-2-[1-(1,2-oxazol-3-ylmethyl)-1H-imidazol-2-yl]quinoline
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(cyclopropylmethyl)piperazine
(4aS,8aS)-2-[2-(dimethylamino)-6-(trifluoromethyl)pyrimidin-4-yl]-decahydro-2,7-naphthyridin-4a-ol
N-[(2,5-difluorophenyl)methyl]-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-amine
methyl 5-{[(2,6-difluorophenyl)methyl]amino}-1-(2-methylpropyl)-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,5S)-1-[(2-fluoro-4-methylphenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
4-{1-azabicyclo[2.2.2]octan-3-yl}-N-(3-ethylphenyl)piperazine-1-carboxamide
N-[(1S,6R)-6-carbamoylcyclohex-3-en-1-yl]-5-(2-chlorophenyl)-2-methylfuran-3-carboxamide
(3S,5R)-1-(3-methylbenzoyl)-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
2-ethyl-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-6-methylpyrimidin-4-amine
(2S)-1-[4-(4-methoxyphenoxy)benzoyl]pyrrolidine-2-carboxamide
3-{[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
8-(1-methanesulfonylpropan-2-yl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(2,3-difluoro-4-methylphenyl)methyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
2-(4-{[(7-chloro-4-methylquinolin-2-yl)(methyl)amino]methyl}piperidin-1-yl)ethan-1-ol
1-[4-(3-methoxyphenyl)phenyl]-N-[2-(pyrazin-2-yl)ethyl]piperidin-4-amine
7-fluoro-3-methyl-N-[2-(methylsulfanyl)ethyl]-1-benzofuran-2-carboxamide
7-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(2S,4R)-4-amino-1-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-N-methylpyrrolidine-2-carboxamide
1'-[2-(2,3-difluorophenyl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-(2-amino-1,3-thiazol-4-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}propanamide
1-(diphenylmethyl)-4-(5-ethyl-1,3-oxazole-4-carbonyl)piperazine
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(methyl)[1-(thiophen-2-yl)ethyl]amine
1-ethyl-8-[3-(5-methylfuran-2-yl)butyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[1-(thiophen-2-yl)propyl]acetamide
(2S,4S)-4-amino-N-ethyl-1-[5-(1H-indol-1-ylmethyl)furan-2-carbonyl]pyrrolidine-2-carboxamide
1-(2-methoxyethyl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-6-oxopiperidine-3-carboxamide
N,N-diethyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-3-amine
1-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(1S)-1-[1-(3-chloro-4-fluorophenyl)-1H-1,2,4-triazol-5-yl]-3-(methylsulfanyl)propyl]acetamide
1-[cyclohexyl(methyl)amino]-3-[3-({[(2-methoxyphenyl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
(1S,5R)-6-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
methyl 1-[(3R,5S)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(4aS,8aR)-6-(5-hydroxypyrazine-2-carbonyl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
4-(1-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carbonyl)morpholine
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
5-{[(2-methanesulfonamidoethyl)carbamoyl]amino}-N,N-dimethyl-1-benzothiophene-2-carboxamide
3-(3-methoxyphenoxymethyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
(1R,3S,5S)-8-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane
1,3-dimethyl-N-[3-(morpholin-4-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
methyl 5-{[(2-chlorophenyl)methyl]amino}-3-(furan-2-amido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[2-(dimethylamino)ethyl]-8-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amino]methyl}phenol