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1-[3-(4-fluorophenoxy)propyl]-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-fluoro-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}benzamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(5-methylpyridine-3-carbonyl)pyrrolidin-3-yl]methanol
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
2-({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}amino)acetamide
1-[2-({[4-(methylsulfanyl)phenyl]methyl}amino)ethyl]-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[3-(diethylamino)pyrrolidin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
1-[(2-methyl-1H-imidazol-4-yl)methyl]-3-[2-(2-methylphenyl)ethyl]piperidine
4-[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]piperazin-2-one
1-{4-[(1-phenylethyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-{[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
N-(2-cyclopropylphenyl)-4-(2-methoxybenzoyl)piperazine-1-carboxamide
3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]urea
4-(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)thiomorpholine
6-(2H-1,3-benzodioxole-5-carbonyl)-3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(4S)-3-[2-(4-methoxyphenoxy)ethyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
1'-(2-propyl-1,3-thiazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]
4-(4-methoxyphenyl)-5-[(2-methylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
5-fluoro-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1H-indole-2-carboxamide
7-(5-chloro-2-methoxyphenyl)-4-cyclobutanecarbonyl-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(3-chloro-4-methoxyphenyl)-4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carboxamide
3-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-4-[(4-methylphenyl)methyl]piperazin-2-one
1-cyclopentyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]piperidine-3-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]ethan-1-one
3-(5-fluoro-2-methoxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
1-acetyl-N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
4-methoxy-3-(morpholin-4-yl)-N-propyl-N-(pyridin-3-ylmethyl)benzamide
3-(3-amino-1H-indazol-1-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-N,N-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1-[4-(furan-2-ylmethoxy)phenyl]-3-methylurea
5-methoxy-3-[2-(1-methylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,3-dimethylbutanamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-(1H-imidazol-1-ylmethyl)piperidine
2-[(3,4-difluorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
2,4-dichloro-3-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}phenol
ethyl 4-({4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazine-1-carboxylate
[(2,4-difluorophenyl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
5-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
7-cyclopropanecarbonyl-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-{[3-(1H-pyrazol-1-yl)propyl]carbamoyl}pyrrolidine-2-carboxylate
5-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
2-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-1,2-oxazolidine
N-methyl-4-(pyrrolidine-1-carbonyl)-6-{thieno[3,2-d]pyrimidin-4-yl}-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
6-(cyclopropylmethoxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
9-(1,4-dioxan-2-ylmethyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(5S,9aS,9bS)-5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one