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N-(1-hydroxybutan-2-yl)-3-(2-methoxyphenyl)-N-(pyridin-3-ylmethyl)benzamide
3-[2-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-5,5-dimethylimidazolidine-2,4-dione
2-phenoxy-N-[4-(4-{[1-(thiophen-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
2-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1,3-benzoxazole
6-methyl-2-phenyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-4-amine
(4aS,7aR)-1-(1,2-oxazole-3-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
1-[(2E)-3-phenylprop-2-en-1-yl]-3-(pyrrolidin-1-yl)piperidine
7-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-(furan-2-amido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-fluoro-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}quinazolin-4-amine
5-chloro-3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-(2-methoxyethyl)-2,5-dimethyl-N-(pyridin-3-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
6-methyl-3-(4-methylpiperazine-1-carbonyl)-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridin-4-one
N-(2-phenylethyl)-6-[(2E)-3-phenylprop-2-en-1-yl]-6-azaspiro[2.5]octane-1-carboxamide
4-[(2-ethoxyphenyl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
dimethyl({4-[4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carbonyl]-1,3-thiazol-2-yl}methyl)amine
(4aS,7aR)-1-[(1-ethyl-1H-indol-6-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(1-acetylpiperidin-4-yl)oxy]-N-[1-(4-fluorophenyl)ethyl]-3-methoxybenzamide
[3-(2-phenoxyethyl)-1-(pyridin-3-ylmethyl)piperidin-3-yl]methanol
1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-methyl-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
N-{[1-(1,3-oxazole-5-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
1-cyclopentyl-4-({[(dimethyl-1,3-thiazol-5-yl)methyl](methyl)amino}methyl)pyrrolidin-2-one
5-{4-hydroxy-1-[(3-methylphenyl)methyl]piperidin-4-yl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1-benzofuran-2-carboxamide
2-(2-ethoxyacetyl)-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-(1-{[5-(2-fluorophenyl)furan-2-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
8-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrazine-2-carbonitrile
N-[(2S,4R,6S)-2-(3-ethoxy-4-methoxyphenyl)-6-(2-methylpropyl)oxan-4-yl]acetamide
3-[2-(2-fluorophenyl)ethyl]-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
3-(4-methyl-1H-pyrazol-1-yl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propan-1-one
(2R,6S)-4-[6-chloro-3-(1H-imidazol-2-yl)imidazo[1,2-a]pyridine-2-carbonyl]-2,6-dimethylmorpholine
4-[(4-chlorophenyl)methyl]-1-(2,5-dimethylpyrimidin-4-yl)piperidine-4-carboxylic acid
3-[(3R,4S)-1-(2-amino-9H-purin-6-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-{[2-(furan-2-yl)-2-oxoacetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
2-(4-{[3-(cyclopentyloxy)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
4-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-1H-pyrazole-3-carboxamide
1-{2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,5S)-6-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}-6-azabicyclo[3.2.1]octane
4-(1-ethyl-1H-imidazol-2-yl)-1-[1-(propan-2-yl)pyrrolidine-3-carbonyl]piperidine
2-[2-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
2-(1H-1,3-benzodiazol-1-yl)-1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}ethan-1-one
3,4-dimethoxy-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
6-amino-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide