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1-(4-methyl-1H-imidazole-5-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-methyl-N-(2-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]morpholin-2-yl}ethyl)but-2-enamide
3-{2-amino-4-methyl-6-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]pyrimidin-5-yl}propanoic acid
1-[(3,4-dimethylphenyl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
3-(2-amino-4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}-6-methylpyrimidin-5-yl)propanoic acid
6-methoxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[4-(ethylamino)pyrimidin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-methoxy-N-(1,4-oxazepan-6-ylmethyl)pyrimidin-4-amine
9-(oxan-2-ylmethyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[4-methoxy-2-(2-methylpropanamido)phenyl]pyrazolo[1,5-a]pyridine-3-carboxamide
5-[1-(2-fluorobenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-{[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]amino}propane-1,2-diol
3-(3-methylpiperidin-1-yl)-1-[4-(pyridin-3-yl)piperazin-1-yl]propan-1-one
N-{1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanamide
4-{2-[4-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]ethyl}morpholine
N-[2-(2,4-difluorophenyl)-1-{1-[(4-hydroxy-3,5-dimethylphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
2-{1-[(2-methylphenyl)methyl]-4-(quinolin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[(1S,5R)-6-(4-methyl-2-phenylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
5-[(2,2-dimethyloxan-4-yl)methyl]-3-(2-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(5-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
N-(2,4-dimethoxyphenyl)-3-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}propanamide
2-[(3-methoxyphenyl)methyl]-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
1-{3-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-4-chlorophenyl}-1H-pyrazole
N-(1-cyclopropylethyl)-5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
4-(benzyloxy)-1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidine
3-[7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-2,3-dihydro-1H-inden-1-one
ethyl 5-(1H-pyrazol-3-yl)thiophene-2-carboxylate
1-[4-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
benzyl({imidazo[1,2-a]pyrimidin-6-ylmethyl})(1,3-thiazol-2-ylmethyl)amine
1-methyl-1'-(oxan-4-yl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
8-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-2-(morpholin-4-yl)ethan-1-one
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-{spiro[2.5]octan-1-ylmethyl}propanamide
N-butyl-2-{methyl[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}acetamide
2-(dimethylamino)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-2,3-dihydro-1H-indene-2-carboxamide
1-methyl-3-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
4-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-2-fluorophenol
6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
8-(3-chlorothiophene-2-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
6-[(3-hydroxypyrrolidin-3-yl)methyl]-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
ethyl 1-[(3-hydroxy-4-methoxyphenyl)methyl]-3-(2-phenylethyl)piperidine-3-carboxylate
2-(3-oxo-1,4-diazepan-1-yl)pyridine-3-carbonitrile
2-methoxy-5-{[methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl})amino]methyl}benzoic acid
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[3-(trimethyl-1H-pyrazol-1-yl)propyl]acetamide
(3R,5S)-5-(3-fluorophenoxymethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
(3S,4R)-1-[(1-ethyl-1H-indol-6-yl)methyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine