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4-hydroxy-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2-[(2-methoxypyrimidin-5-yl)formamido]-N-(2-methylphenyl)acetamide
(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)(1,3-thiazol-2-ylmethyl)amine
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-(4-phenyl-1,4-diazepan-1-yl)propan-1-one
5-chloro-4,6-dimethyl-2-oxo-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
3-(2-chlorophenyl)-1-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]propan-1-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-(2,3-dihydro-1-benzofuran-7-yl)-N-methylpyridine-3-carboxamide
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-cyclohexyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
N-(1-methanesulfonylpiperidin-4-yl)-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-[2-(pyrimidin-2-ylsulfanyl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
dimethyl(3-{2-[1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
2-{3-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-imidazol-2-yl]phenoxy}acetamide
N-{2-[7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclohexanecarboxamide
2-(4-{6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}-6-methylpyrimidin-2-yl)phenol
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
1-(6-{6-[3-(dimethylamino)propoxy]pyridin-3-yl}-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
[2-(3-chlorophenyl)ethyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-acetamidopropanamide
3-(3-ethynylbenzoyl)-9-methoxy-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-{1-[(2-chloro-6-fluorophenyl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl}piperidin-2-one
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-methoxyphenyl)ethyl]acetamide
1-(1,3-oxazole-5-carbonyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(4,5-dimethyl-3-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}thiophen-2-yl)-1H-1,2,3,4-tetrazole
6-(cyclopropylmethoxy)-4-(furan-3-carbonyl)-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
7-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3H,4H-pyrido[3,4-d]pyrimidin-4-one
1-{1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}-2-methylpiperidine
1-methyl-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(propan-2-yl)-5-[2-(thiophen-2-yl)-1,3-thiazol-4-yl]-1,2,4-oxadiazole
methyl 2-{4-[(piperidin-3-yl)amino]piperidin-1-yl}acetate
methyl 6-(1-benzofuran-2-carbonyl)-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-4,6-dimethylpyrimidin-2-amine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(pyridin-3-yl)acetamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[(1s,5s)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecan-3-yl]ethan-1-one
ethyl 1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-imidazole-2-carboxylate
N-(1-{1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
2-{[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}benzoic acid
(4aS,8aR)-6-[(4-fluoro-2-methylphenyl)methyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(1-benzylpiperidin-4-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)-N-methylacetamide
N-[(3S,4R)-1-(3,4-dimethoxybenzenesulfonyl)-4-propylpyrrolidin-3-yl]acetamide
N,N,4-trimethyl-3-({[2-(1H-pyrazol-4-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4-(1H-1,2,4-triazol-1-yl)butanamide
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-[4-(difluoromethoxy)-2-methylphenyl]urea
N,N-diethyl-1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
3-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]propanamide
4-oxo-4-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]butane-1-sulfonamide
3-(oxan-4-yl)-5-(1H-pyrazol-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
(2S,4R)-1-benzyl-4-{[(2,4-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide