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N-[(3-chlorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[5-(pyrrolidine-1-carbonyl)furan-2-yl]-1H-imidazole-4-carboxylic acid
(3aS,6aS)-2-acetyl-5-[(4-methylphenyl)methanesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(4-chlorophenyl)methyl]-N-[2-(4-fluorophenoxy)ethyl]-6-oxopiperidine-3-carboxamide
1-(1-methyl-1H-imidazol-2-yl)-2-[(6-phenylpyridazin-3-yl)amino]ethan-1-ol
6-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
N-[3-(1H-indol-1-yl)propyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1S,4S)-2-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)-2-azabicyclo[2.2.1]heptane
1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]-4-(oxolan-2-ylmethyl)piperazine
2-methoxy-1-{4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl}ethan-1-one
N-[2-methyl-1-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]methanesulfonamide
7-(2-methoxyethyl)-2-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
4-(1-tert-butyl-1H-pyrrole-3-carbonyl)-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]pyridine-4-carboxylic acid
3-(2,6-difluorobenzoyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-{4-[4-(4-benzylpiperidine-1-carbonyl)phenoxy]piperidin-1-yl}-2-methoxyethan-1-one
[(3R,4S)-1-{[4-(2-aminoethyl)phenyl]methyl}-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methyl-2-phenylpiperazine
2-(cyclopropylmethyl)-9-(trimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-({2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}amino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-(naphthalen-1-yl)piperidine-1-carboxamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
3-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-cyclopentyl-1,4-diazepane
(1S,6R)-3-methyl-4-oxo-N-(4-phenylphenyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N-(1-{7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,5-difluorobenzamide
7-[(4-hydroxy-2,6-dimethylphenyl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N1-(3-chloro-4-propoxyphenyl)-N2-methylpyrrolidine-1,2-dicarboxamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(2H-indazol-2-yl)ethan-1-one
2-[4-(1,7-dimethyl-1H-indole-2-carbonyl)piperazin-1-yl]-1,3-benzoxazole
6-(cyclobutylamino)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
(2E)-1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
6-[(dimethylamino)methyl]-N-(2,3-dimethylphenyl)-1,4-oxazepane-4-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]acetamide
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-cyclopentyl-6-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(3-{2-[1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}but-3-en-1-one
8-(3-methoxy-2-methylbenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]propan-1-ol
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2-phenylethyl)pyrrolidin-3-yl]methanol
2-(2-chlorophenyl)-2-{[1-(furan-2-ylmethyl)piperidin-4-yl]formamido}acetic acid
N-[(3S,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-ethyl-1H-pyrazole-5-carboxamide
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-2-(1H-1,2,4-triazol-1-yl)acetamide
5-[3-(piperidin-1-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(pyridin-4-yl)propanamide
(1S,5R)-3-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(cyclohexylmethyl)-5-(2,3,4-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole