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N-cyclooctyl-5-(3-methylpiperidine-1-carbonyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
1-cyclopentyl-N5-ethyl-N3-methyl-N3-[2-(4-methylphenoxy)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(1-benzothiophen-5-ylmethyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}propanoic acid
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
3-[2-oxo-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
3-{[5-(1-benzyl-1H-imidazol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}urea
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-(4-methoxynaphthalen-1-yl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
4-({4-[2-(2-ethylpiperidine-1-carbonyl)-4-methylphenoxy]piperidin-1-yl}methyl)pyridine
N-[4-(4-{[2-(morpholin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]-5-phenylpentanamide
5-({[(3-{2-[4-(2,3-dimethyl-1H-indole-7-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-methyl-1H-imidazole-2-carboxamide
N-benzyl-N,1-dimethyl-5-[(pyridin-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1H-pyrazol-3-one
3-chloro-N-[2-(dimethylamino)ethyl]-4-[(1-propylpiperidin-4-yl)oxy]benzamide
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-9H-fluorene-9-carboxamide
1-(2,3-dimethoxyphenyl)-2-(3-fluorobenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
3-[3-(2-methoxyphenoxy)propyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
3-methyl-5-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}-1H-1,2,4-triazole
methyl (2S)-1-[(4-{[2-(2-methoxyphenyl)ethyl]amino}quinazolin-2-yl)methyl]pyrrolidine-2-carboxylate
{3-[(2,4-difluorophenyl)methyl]-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-yl}methanol
(2S)-2-({2,7-dimethylpyrazolo[1,5-a]pyrimidin-5-yl}formamido)-3-(4-hydroxyphenyl)propanamide
N-cyclopentyl-2-hydroxy-N-(3-phenylprop-2-yn-1-yl)benzamide
N-[3-(furan-2-yl)propyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
(3S,5R)-1-(3-methylfuran-2-carbonyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(3-methyl-1,2-oxazol-5-yl)acetamide
3-{2-amino-4-methyl-6-[methyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})amino]pyrimidin-5-yl}propanoic acid
4-methyl-N-[3-methyl-2-(pyrrolidin-1-yl)butyl]-3-phenyl-1H-pyrazole-5-carboxamide
1-ethyl-N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(propoxycarbonyl)piperidine-4-carboxylic acid
5-(3-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)-5-(thiophen-3-ylmethyl)pyrrolidin-2-one
1-methyl-4-[2-(4-phenyl-1H-imidazol-5-yl)phenyl]piperazine
7-fluoro-1-methyl-2-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-[(3-ethoxyphenyl)methyl]-6-ethyl-N-(2-hydroxyethyl)-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[(1-ethylpyrrolidin-3-yl)methyl]-1-[4-(propan-2-yl)phenyl]urea
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(propan-2-yl)urea
N-cyclohexyl-3-(4-hydroxyphenyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
5-acetyl-N-[2-(2-chlorophenyl)-2-hydroxyethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl](quinolin-4-ylmethyl)amine
5-(1-tert-butyl-5-oxopyrrolidine-3-carbonyl)-N-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
2-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazin-1-yl}-1,3-benzothiazole
(4aS,8aR)-6-(2-aminopyridine-4-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-benzyl-N-[(1-ethylpiperidin-3-yl)methyl]-N,1-dimethyl-5-propanamido-1H-1,3-benzodiazole-7-carboxamide
dimethyl({4-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]phenyl}methyl)amine
3-[1-(6-methyl-4-oxo-4H-pyran-2-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide