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1-benzyl-2-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
3-[2-(dimethylamino)ethyl]-5-{1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
4-(dimethyl-1,2-oxazol-4-yl)-2-(methylsulfanyl)pyrimidine
N-[(3S,4R)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
4-(piperidin-3-ylmethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
N,8-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
3-(azocan-1-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]propanamide
4-{[3-(4-phenoxybenzoyl)piperidin-1-yl]methyl}pyridine
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
1-(5-methoxy-2-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
N-(2,2-difluoroethyl)-6-(2,5-dimethylfuran-3-yl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyridine-2-carboxamide
2-methyl-6-{[1-methyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}heptan-2-ol
2-[6-(morpholin-4-yl)pyrimidin-4-yl]benzonitrile
N-{1-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]piperidin-4-yl}acetamide
[7-chloro-5-(2,4-dimethoxypyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-[4-(2H-1,3-benzodioxol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
6-[4-(6-oxo-2-phenyl-1,6-dihydropyrimidin-4-yl)piperidin-1-yl]pyridine-3-carbonitrile
3-ethyl-8-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-methyl-1,3-benzothiazol-5-yl)-6-[2-(pyrimidin-2-ylsulfanyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
methyl 5-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
2-[(5-methylpyrazin-2-yl)methyl]-8-[(6-methylpyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(hydroxymethyl)-9-(pyridin-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(1H-imidazol-1-yl)ethan-1-one
N-[(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
1-(cyclohexylmethyl)-6,7-dimethoxy-3-(morpholin-4-ylmethyl)-1,2-dihydroquinolin-2-one
4-hydroxy-N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(2-hydroxyethyl)-1,3-oxazole-4-carboxamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
5-(2,4-dimethylbenzoyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}urea
methyl 6-cyclohexanecarbonyl-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)quinolin-8-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-phenoxyacetamide
4-methyl-5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
2-(pyridin-2-ylmethyl)-9-(thiophene-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R)-2-amino-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)propanamide
2-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-butyl-1-methyl-4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazin-2-one
1-methyl-2-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
2-methyl-4-{3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}but-3-yn-2-ol
2-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
2-(4-fluorophenyl)-N-[2-methyl-4-(methylcarbamoyl)phenyl]piperidine-1-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(4-fluoro-3-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(1-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-methylfuran-3-carboxamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2,4-dimethoxyphenyl)ethan-1-one
{[6-(6-fluoroquinolin-8-yl)pyridin-3-yl]methyl}dimethylamine
(3R,4R)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
(1S,5R)-3-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one