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N-[2-(3-chlorophenyl)ethyl]-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-ethyl-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1,2-oxazole-4-carboxamide
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-{[2-(methylsulfanyl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
N-[2-(1-{[(2-chlorophenyl)carbamoyl]carbonyl}piperidin-2-yl)ethyl]acetamide
3-(2-fluorophenyl)-6-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
6-{2-[(6-methoxypyrimidin-4-yl)amino]ethyl}-2-methylpyrimidin-4-ol
1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-amine
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-(1-methylcyclopropanecarbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-5-fluoro-N,N-dimethylpyrimidin-4-amine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-[(1S,5R)-6-[4-(pyrrolidin-1-ylmethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
methyl 7-oxo-3-(quinolin-2-ylmethyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1-propyl-1H-pyrazole
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanamide
1-[4-(morpholine-4-carbonyl)phenyl]-N-[3-(pyridin-3-yl)propyl]piperidin-4-amine
N-[2-({5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethyl]acetamide
8-(3-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(4-fluorophenyl)propanoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-[3-(trifluoromethyl)phenoxy]piperidine
6-fluoro-2-oxo-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(3-phenylpropyl)-8-(1,3-thiazol-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
3-[(cyclopentylamino)methyl]-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}hexan-1-one
methyl (2S)-2-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamido)-3-methylbutanoate
1-{1-[(3-methyl-1-benzofuran-2-yl)methyl]azetidin-3-yl}piperidine
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-{4-[1-(2-methoxyacetyl)piperidine-3-carbonyl]piperazin-1-yl}benzonitrile
N-[(5-fluoro-2-methylphenyl)methyl]-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
[1-({4-[3-(5-methylfuran-2-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-2-yl]methanol
(3aS,6aS)-2-(oxan-4-yl)-5-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 3-(2-chlorobenzenesulfonamido)-5-[(phenylformamido)methyl]benzoate
{2-[3-(trifluoromethyl)phenyl]pyridin-4-yl}methanol
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
1-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]ethyl}-1H-indazole
1-(cyclopent-3-ene-1-carbonyl)-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-6-ol
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
5-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
2,3-dimethoxy-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}benzamide
3-(2-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-benzyl-N-[2-(dimethylamino)ethyl]-1-(methoxymethyl)cyclopropane-1-carboxamide
4-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-N,N-dimethylpiperazine-1-carboxamide
2-cyclopropyl-5-{[(2S,5R)-5-[(4-methylpiperazin-1-yl)methyl]oxolan-2-yl]methyl}-1,3-benzoxazole
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-(2-methoxyphenoxy)azetidine
N-[(2,6-dimethoxyphenyl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
5-[2-(3-hydroxy-1,2-oxazol-5-yl)ethyl]-3-(4-methoxyphenyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-[2-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)-4-(pyrimidin-2-yl)phenoxy]acetic acid
5,6-dimethyl-3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one