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(2S,4S)-N-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-4-(furan-2-amido)pyrrolidine-2-carboxamide
N-({1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-4-(2,6-dimethylpyridin-4-yl)piperazine
2-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-N-(5-methyl-1,2-oxazol-3-yl)-2-oxoacetamide
3-(4-chlorobenzoyl)-1-[(2,3-dimethoxyphenyl)methyl]piperidine
methyl 3-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-5-[3-(trifluoromethyl)benzamido]benzoate
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-methylpiperidine
1-{1-ethyl-5-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-phenylpiperazine
5,7-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-benzothiazole-6-carboxamide
2-(4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
1-[(3S)-3-ethylmorpholin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethan-1-one
1-[1-(4-chloro-3-fluorobenzoyl)piperidin-4-yl]piperidin-3-ol
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(1R)-1-phenylethyl]pyrimidin-2-amine
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(3S,4R)-1-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
2,3-dimethyl-6-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
2-(5-{3-[2-(4-methylpiperazin-1-yl)ethyl]-1,2,4-oxadiazol-5-yl}-1H-pyrazol-3-yl)phenol
dimethyl[2-({1-[(6-methylquinolin-5-yl)methyl]piperidin-4-yl}oxy)ethyl]amine
4-[2-(4-methylpentyl)morpholin-4-yl]-4-oxobutanamide
6-methyl-5-{5-[2-(morpholin-4-yl)pyridin-3-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
2-ethoxy-5-(2-{[(1S)-1-(3-methylpyridin-2-yl)ethyl]amino}pyrimidin-4-yl)benzoic acid
N-cyclopentyl-3-{[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]sulfamoyl}benzamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N-methylpiperidine-2-carboxamide
1-[2-(1-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
1-(4-benzylpiperazin-1-yl)-3-(1-methanesulfonylpiperidin-3-yl)propan-1-one
7-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-[(3S,4R)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-methyl-1-(6-methylpyridine-3-carbonyl)-N-(2-phenylethyl)piperidin-3-amine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
1-{2-[(5-ethyl-2-methylpyrimidin-4-yl)amino]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
(4aS,8aR)-2-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)-decahydroisoquinoline
N-[(4-methylphenyl)(pyridin-4-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
(2S,4R)-4-amino-N-methyl-1-(2-phenylquinoline-4-carbonyl)pyrrolidine-2-carboxamide
3-{7-ethyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-N-[(4-methylphenyl)methyl]propanamide
5-acetyl-3-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
ethyl 1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
3-[(3,5-dimethylphenyl)methyl]-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
4-cyclopentyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine
N-[2-methyl-2-(morpholin-4-yl)propyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[(4-fluorophenyl)methyl]-N-methyl-5-propyl-1,3,4-oxadiazol-2-amine
[1-(4-methoxypyrimidin-2-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
[(3R,4R)-1-(5-chloro-2-methoxybenzoyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-[2-(2,4-difluorophenyl)ethyl]-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
N-(4-chloro-2-methylphenyl)-3-(dimethylamino)piperidine-1-carboxamide
2-[3-(5-methyl-1H-indol-3-yl)phenoxy]acetamide
2-[4-(1H-indol-2-ylmethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol