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N-[(2R,3R)-2-methoxy-1'-(quinolin-6-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
(1R,7S)-N-methyl-4-oxo-3-(pentan-3-yl)-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-chloro-6-methoxy-4-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenol
(3S,9aR)-8-(2,5-dimethylbenzenesulfonyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{5-[(1R)-1-phenylpropyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-(ethylsulfanyl)propanamide
2-{[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]amino}-N-(pyrazin-2-yl)acetamide
5-{1-[(2-chloro-6-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}-2,2-dimethylthiomorpholin-3-one
N-(pyridin-2-ylmethyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-({7-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
{3-[(2,4-difluorophenyl)methyl]-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}methanol
2-[2-(dimethylamino)ethyl]-9-[5-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
({5-[1-(cyclopentylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
ethyl 1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-3-(2-phenoxyethyl)piperidine-3-carboxylate
(3aR,7aS)-2-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(2-methylphenyl)ethan-1-one
4-[(4-fluorophenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
9-(cyclopropylmethyl)-4-(1H-imidazol-4-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-benzyl-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2E)-1-[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(2-fluorophenyl)ethyl)piperidin-1-yl]-2-methylbut-2-en-1-one
methyl 4-methyl-2-{2-[4-(pyridin-4-yl)-1,4-diazepan-1-yl]acetamido}-1,3-thiazole-5-carboxylate
6-methyl-2-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
4-({4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]furan-2-yl}methyl)morpholine
1-acetyl-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)piperidine-4-carboxamide
(5Z)-5-{2-[6-(benzyloxy)-4-cyclohexyl-3-oxo-1,4-diazepan-1-yl]-2-oxoethylidene}-1,3-thiazolidine-2,4-dione
2-[1-(furan-3-ylmethyl)-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-2-yl]ethan-1-ol
5-acetyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)thiophene-3-carboxamide
6-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-methyl-N-(2-methylpropyl)-N-(thiophen-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-[(1-benzylpyrrolidin-3-yl)methyl]-4H-1,2,4-triazole
4-{3-[4-(3,4-dimethylphenyl)-1H-1,2,3-triazol-1-yl]propyl}pyridine
8-[(3-hydroxyphenyl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(cyclopent-3-en-1-yl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
(3R,5R)-5-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidine-1-carbonyl]pyrrolidin-3-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-methoxycyclohexanecarbonyl)piperidin-3-ol
3-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-phenyl-1-(4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)ethan-1-ol
2-(4-hydroxyphenyl)-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-(2-methoxyphenyl)-4-[(pentan-3-yl)amino]pyrrolidin-2-one
(3S,4S)-3-hydroxy-4-{[(4-{[2-(2-methoxyphenyl)ethyl]amino}quinazolin-2-yl)methyl](methyl)amino}-1λ6-thiolane-1,1-dione
4-methoxy-N-{[1-(3-phenoxypropanoyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
2-[4-({methyl[(1-methylpiperidin-4-yl)methyl]amino}methyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
(3S,4S)-N-ethyl-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carboxamide
7-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
2-benzyl-N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-1,3-thiazole-4-carboxamide
2-(2-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1-(difluoromethyl)-1H-pyrazole-3-carboxamide