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N-{1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-{4-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]benzoyl}piperidine
1-(cyclopentylcarbamoyl)-4-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepane-6-carboxylic acid
5-methyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-(4-methylpent-3-en-1-yl)piperidin-2-one
9-(cyclopropylmethyl)-1-methyl-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazole-3-carboxamide
5-{3-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1,3,4-thiadiazol-2-amine
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-4-[(2-hydroxyethyl)(methyl)amino]benzamide
3-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one
(3aR,6aR)-2-(2,4-dimethylbenzoyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine-3-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
2-methyl-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-N,N-diethylpiperidine-4-carboxamide
methyl 3-acetamido-5-[(2-ethylbutyl)amino]-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{1-[3-(1H-imidazol-1-yl)propanoyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethan-1-one
8-[2-(3-methoxyphenoxy)ethyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(ethanesulfonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
4-(1-hydroxy-2-methylpropyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
N-methyl-2-(1-methyl-1H-indol-3-yl)-N-[1-(pyridin-2-yl)propan-2-yl]acetamide
2-amino-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]ethan-1-one
2-(3-hydroxypiperidin-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}acetamide
methyl 4-{5-chloro-2-[(3-acetamidopropanamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
4-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
2-(2-methoxyethyl)-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(2-acetamidoethyl)propanamide
2-[5-(1-ethyl-1H-pyrazol-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]-6-methylpyridine
6-(2-aminoethyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-methylpyrimidin-4-amine
(4aS,7aR)-1-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-1,2,3,4-tetrahydroisoquinoline
1-[2-(2,5-dimethoxyphenyl)ethyl]-N,N-dimethylpyrrolidin-3-amine
7-(2-cyclohexylethyl)-2-(1H-imidazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(2-hydroxybutyl)benzamide
2,4-difluoro-3-methoxy-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)benzamide
1-(4-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-3-methylphenyl)-1H-pyrazole
N-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[2-(oxan-2-yl)ethyl]amine
1-[(4-chlorophenyl)methyl]-6-oxo-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
methyl 5-oxo-5-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)pentanoate
3-{1-methyl-5-[1-(4-methylphenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
9-methoxy-4-[5-(methoxymethyl)furan-2-carbonyl]-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-1-tert-butyl-5-oxopyrrolidine-3-carboxamide
3-hydroxy-3-[({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)amino)methyl]-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
2-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-3,5-dimethyl-1H-indole
(1S,2R,3R,4R)-N2-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-N3-cyclopropylbicyclo[2.2.1]hept-5-ene-2,3-dicarboxamide