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N,N-dimethyl-6-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidin-4-amine
N-ethyl-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]furan-2-carboxamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-2-ylsulfanyl)propan-1-one
N,1-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-3-(thiophen-2-yl)-1H-pyrazole-5-carboxamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-(2-methylbenzoyl)piperidine-3-carboxylate
3-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-1-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}urea
4-[(2-fluoro-5-sulfamoylphenyl)formamido]-N,4-dimethylpentanamide
N-(4-methylphenyl)-2-[(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)amino]propanamide
(8R,9aS)-8-hydroxy-2-(2-methylprop-2-en-1-yl)-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
1-cyclopentyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-6-oxopiperidine-3-carboxamide
4-[1-(3-methylbutyl)-5-[2-(methylsulfanyl)pyridine-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
5-[1-(benzenesulfonyl)cyclopropanecarbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
2-benzyl-8-[3-(4H-1,2,4-triazol-4-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
14-[4-ethoxy-3-(hydroxymethyl)phenyl]-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4-(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)pyridine
2-ethoxy-5-(2-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
methyl 2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butanoate
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
{1-[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]cyclopentyl}methanol
N-{3-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]phenyl}acetamide
N-[(5-methylpyrazin-2-yl)methyl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
3-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
2-[4-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-6-methylpyrimidin-2-yl]phenol
N,N,5-trimethyl-2-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}pyrimidin-4-amine
N-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
(1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)methanamine
4-methyl-N-(prop-2-en-1-yl)-N-(propan-2-yl)-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
N-[1-(4-fluorophenyl)piperidin-4-yl]-3-(1-methylpiperidin-2-yl)propanamide
4-(azepan-1-ylmethyl)-N-[2-(2-hydroxyethyl)phenyl]benzamide
1-{3-[2-(4-methylpentyl)morpholin-4-yl]-3-oxopropyl}azepan-2-one
2,5-dimethyl-3-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrazine
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
3-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-1-ol
(3aS,6aS)-2-methyl-5-(1,3-thiazol-5-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
{4-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenyl}methanol
3-(3-fluorophenyl)-4-[(8-methylquinolin-5-yl)methyl]piperazin-2-one
methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})(1,2-oxazol-5-ylmethyl)amine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})(thiophen-2-ylmethyl)amine
2-(1-cyclohexyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1-(3,4-dimethoxyphenyl)ethan-1-amine
(3S)-1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-ol
N-(cyclohex-1-en-1-ylmethyl)-2-[3-(1H-imidazol-1-yl)propyl]-1-oxo-2,3-dihydro-1H-isoindole-5-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[4-(ethylamino)pyrimidin-2-yl]pyrrolidin-3-yl]methanol