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(1S,5R)-3-[(2-fluorophenyl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
N5-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-N3,N3-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(3-hydroxy-3-methylbutyl)-N-(pyridin-4-ylmethyl)benzamide
1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}-1,4-diazepan-6-ol
[(3R,4R)-1-(3-fluorobenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazole
ethyl 3-(2-phenoxyethyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine-3-carboxylate
7-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepan-5-one
N-({8-[(2,6-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butan-1-one
6-tert-butyl-N-[(2-methoxyphenyl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N3-[2-(2-ethylphenoxy)ethyl]-N3-methylpiperidine-1,3-dicarboxamide
3-fluoro-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
(2S,4S,5R)-4-[(carboxymethyl)carbamoyl]-2-ethyl-5-(4-fluorophenyl)-1-methylpyrrolidine-2-carboxylic acid
N-(3,5-dimethylphenyl)-2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
1-[1-({1-[(8-fluoroquinolin-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
(2S)-4-methyl-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-2-phenylpiperazine
2-(3-fluorophenoxymethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-methyl-4-[4-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenyl]butan-2-ol
5-amino-3-[5-(oxan-2-yl)furan-2-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-2-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
3-[(benzylamino)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
2-[(4aR,7aS)-4-(3-fluorobenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2,4-dimethyl-N-[2-(4-sulfamoylphenyl)ethyl]pyrimidine-5-carboxamide
N2-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
1-({3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
N-{1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl}acetamide
2-[2-oxo-4-(2-propylpentanoyl)piperazin-1-yl]benzonitrile
N3-cyclopropyl-1-[(3-methoxyphenyl)methyl]-N5-[(4-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]propanamide
(3aS,6aR)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 7-oxo-3-[3-(prop-2-en-1-yloxy)benzoyl]-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(1H-pyrazol-1-ylmethyl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]benzamide
(isoquinolin-5-ylmethyl)(methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
2-(2H-indazol-2-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[3-(dimethylamino)propyl]-5-[(3-fluorophenyl)methyl]-5-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(2S)-2-amino-3-phenyl-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
4-[5-({cyclopropyl[(2-methoxyphenyl)methyl]amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
2-(2H-1,3-benzodioxol-5-yl)-1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1H-imidazole
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(2,6-difluorophenyl)methyl]piperidine
N-{3-[(3S)-3-ethylmorpholin-4-yl]-3-oxopropyl}-N-methylmethanesulfonamide
6-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyridazin-3-amine
2-cyclopropyl-4-methyl-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrimidine
2-(3,4-dichlorophenyl)-4-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]morpholine
ethyl 1-[3-(1H-imidazol-2-yl)benzoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate