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N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N,2,2-trimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
3-(6-methoxypyridin-3-yl)-1-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)urea
1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(thian-4-yl)piperazine
1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
N-[(3S)-1-benzylpiperidin-3-yl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-{1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-[4-(furan-2-yl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
4-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-1,2,3-triazole
1-ethyl-N-[(5-fluoro-2-methylphenyl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{2-[2-(dimethylamino)ethyl]piperidine-1-carbonyl}-1-ethyl-1,2-dihydropyridin-2-one
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N5-cyclopentyl-N6-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(1H-pyrazol-3-ylmethyl)amine
3-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-5-(propan-2-yl)-1,2-oxazole
2-({2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetamido}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-[(2,4-difluorophenyl)methyl]-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[methyl(piperidin-4-yl)amino]-N,N-bis(1,3-oxazol-4-ylmethyl)acetamide
3-(1-{2-[3-chloro-4-(propan-2-yloxy)phenyl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 2-{1-[4-(2-oxopyrrolidin-1-yl)benzoyl]piperidin-2-yl}acetate
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
1-{3-[(cyclobutylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(3R,4S)-4-[({2,4-dimethyl-5-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)(methyl)amino]oxolan-3-ol
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-[2-(2-fluorophenoxy)ethyl]pyrimidine-5-carboxamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)oxane-4-carboxamide
N-[2-(diethylamino)ethyl]-2-{1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-methylacetamide
2-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
(3S,4S)-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
3-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)propan-1-ol
6-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidine-1-carbonyl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
7-chloro-3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-4-phenylbutane-1,2-dione
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
3-methyl-N-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
2-(2,4-dimethylphenyl)-2-(4-{[(propan-2-yl)carbamoyl]methyl}piperazin-1-yl)acetic acid
5-(2-chloro-4-methoxyphenoxymethyl)-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-methanesulfonamidoacetamide
2-(2-cyclopentylacetyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,9S)-11-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-[({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
1-benzyl-N-(cyclopropylmethyl)-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide