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2-(methylamino)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}benzamide
(2E)-1-{3-[5-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
N-(cyclohexylmethyl)-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetamide
4-(1-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidin-4-yl}azetidin-3-yl)morpholine
6-methoxy-3-methyl-N-[1-(pyrrolidin-1-yl)propan-2-yl]-1-benzofuran-2-carboxamide
4-[(2-methylpyridin-3-yl)oxy]-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-4-carboxylic acid
5-{1-[4-(furan-2-yl)benzoyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(3-chlorophenyl)propanamide
2-(2-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
8-(6-methyl-2-propylpyrimidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)acetamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N,5-dimethyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
(1S,5R)-6-methyl-3-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
5-methyl-2-[4-(methylsulfanyl)phenyl]-4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1,3-oxazole
1-[cyclohexyl(methyl)amino]-3-[3-({[3-(pyridin-3-yl)propyl]amino}methyl)phenoxy]propan-2-ol
5-[2-(1H-pyrazol-4-yl)ethyl]-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
8-(2-aminoethyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-phenyl-1-(1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidin-4-yl)ethan-1-ol
8-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 6-[(2,5-dimethylphenyl)methyl]-2-(thiomorpholine-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(4-ethylphenyl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
(3R,4S)-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-3,4-dimethylpiperidin-4-ol
3-({[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino}methyl)piperidin-3-ol
3-(1H-imidazol-2-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-methyl-1-(3-methylphenyl)piperazin-2-one
4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-hydroxy-3-methoxypropyl)-3-methoxybenzamide
1-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
benzyl(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(3R,4R)-4-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)piperidin-3-ol
2-[4-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-4-(propan-2-yl)-6-(trifluoromethyl)pyrimidine
N-(4-fluorophenyl)-1-(5-methyl-1H-indole-2-carbonyl)piperidin-3-amine
3-[({[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}amino)methyl]piperidin-3-ol
2-(2-hydroxyethyl)-9-(1H-indole-6-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-methanesulfonyl-1'-[(2R)-oxolane-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(5-ethylfuran-2-yl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-methoxy-1-(pyridin-2-yl)ethyl]acetamide
4-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}-6-(2-methylpropyl)pyrimidin-2-amine
1-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-(pyridin-2-yl)ethan-1-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1,2-oxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-[1-tert-butyl-5-(morpholin-4-ylmethyl)-1H-1,2,4-triazol-3-yl]benzamide
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidine
(1R,3S)-7-(4-aminopyrimidin-2-yl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-N-[(2-methylphenyl)methyl]acetamide
(oxolan-2-ylmethyl)({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})(thiophen-3-ylmethyl)amine
methyl 2-[4-(but-3-en-1-yl)-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetate