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4-[1-(7-fluoroquinazolin-2-yl)piperidin-4-yl]-1,4-oxazepan-6-ol
methyl 5-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
3-{2-oxo-2-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethyl}-1,3-oxazolidin-2-one
(1S,3R)-3-(2-ethoxyacetamido)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]cyclopentane-1-carboxamide
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyrazin-2-yl)ethyl]pyridin-2-amine
N-benzyl-N-ethyl-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
methyl 1-methyl-3-(3-phenylpropanamido)-5-{[(2,3,4-trimethoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-2-cyclopentyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
9-(2-aminopyrimidin-4-yl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
4-{4-[(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)methyl]phenyl}-2-methylbutan-2-ol
1-(furan-2-ylmethyl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}piperidin-4-amine
ethyl[(2E)-3-(furan-2-yl)prop-2-en-1-yl]{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
7-(4-fluorophenyl)-2-[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{thieno[2,3-d]pyrimidin-4-yl}piperazin-2-one
1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-(dimethyl-1,3-oxazole-5-carbonyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
N-cyclopropyl-2-[3-(4-phenylbenzoyl)piperidin-1-yl]acetamide
4-ethyl-3-({1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[(2S,4R)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidin-1-yl]methyl}phenol
3-[(benzylsulfamoyl)amino]-N-(2-fluoro-4-methylphenyl)propanamide
5-(furan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-ethylpyrimidine-5-carboxamide
2-(dimethylamino)-1-(4-hydroxypiperidin-1-yl)-2-(2-methylphenyl)ethan-1-one
3-[(3R,4S)-1-(4-methyl-1,3-thiazole-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
6,7-dimethyl-2-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1H-1,3-benzodiazole
3-(2-phenoxyethyl)-8-(thiolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-4-(1-methylpiperidin-4-yl)piperidine
(4aS,7aR)-1-(2-hydroxyacetyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl({[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})(thiophen-3-ylmethyl)amine
N-cyclopropyl-4-methoxy-3-{[(1H-pyrazol-3-ylmethyl)carbamoyl]amino}benzamide
11-{[(3,4-difluorophenyl)methyl]amino}-4-[2-(morpholin-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-{[2-(pyrrolidine-1-sulfonyl)ethyl]amino}-N-(1,3-thiazol-2-yl)propanamide
4-(4-{[(4-methoxyphenyl)methyl]amino}piperidin-1-yl)-N-(1-phenylethyl)benzamide
(3S,4R)-4-(hydroxymethyl)-1-(pyridin-2-ylmethyl)piperidin-3-ol
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
4-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
(2S,4S)-4-amino-1-[(2S)-2-(6-methoxynaphthalen-2-yl)propanoyl]-N-methylpyrrolidine-2-carboxamide
(1S,6R)-3-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
1-{5,7-dimethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carbonyl}piperidine-4-carbonitrile
3-{4-[1-(4-chlorophenyl)cyclobutanecarbonyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
methyl (1R,3S,3aR,6aS)-5-methyl-3-[3-(morpholin-4-ylmethyl)phenyl]-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-[2-(2,2-diethylmorpholin-4-yl)-2-oxoethyl]-4-(furan-3-ylmethyl)piperazin-2-one
7-(cyclopropylmethyl)-2-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylamino)ethan-1-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
1-(butane-1-sulfonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2,2,2-trifluoroethyl)acetamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-[(1H-indol-3-ylmethyl)amino]pyrrolidine-2-carboxamide