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1-ethyl-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1,9-dimethyl-4-[3-(2-methylphenyl)benzoyl]-1,4,9-triazaspiro[5.5]undecane
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]-3-ethyl-1,2-oxazole-5-carboxamide
2-{4-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]piperazin-1-yl}-3-methylpyrazine
N-ethyl-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-4-(methylsulfanyl)benzamide
8-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(2-hydroxyethyl)-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-(1,3-thiazol-2-ylmethyl)butanamide
methyl 6-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyridine-2-carboxylate
N-[4-({[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]acetamide
9-methyl-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-9H-carbazole-3-carboxamide
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]azepane
1-(4-chlorophenyl)-3-(1,4-dioxan-2-ylmethyl)urea
(3-{2-azabicyclo[2.2.1]hept-5-en-2-yl}propyl)({[7-chloro-2-(2,3-dimethoxyphenyl)quinolin-3-yl]methyl})amine
N-[(2S)-1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl]acetamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
(3S)-1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-N,N-dimethylazepan-3-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
N-(2-{5-[(2E)-but-2-en-2-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyridine-3-carboxamide
5-fluoro-N4,N4-dimethyl-N2-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrimidine-2,4-diamine
1-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]urea
2-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(thiophen-2-ylformamido)propanamide
N-{2-[7-(2-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-3-carboxamide
4-chloro-N,1-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
4-phenyl-2-{4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}pyrimidine
2-methyl-1-(pyrrolidin-3-ylmethyl)-1,4-dihydroquinolin-4-one
5-[(3-methoxyphenyl)methyl]-N-[(4-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2,3-dihydro-1H-inden-1-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(1H-pyrrole-3-carbonyl)piperazin-2-one
4-{4-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]phenyl}-2-methylbutan-2-ol
1-methyl-8-{[3-(5-methylfuran-2-yl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(4-tert-butylphenyl)-6-(methoxymethyl)pyrimidine
N-{2-[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-(4-fluorophenyl)acetamide
N,N-dimethyl-2-(2,3,4-trimethoxyphenyl)pyrimidin-4-amine
3-[1-(6-cyanopyridine-3-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
7-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
4-(2,5-dihydro-1H-pyrrol-1-yl)-7-(piperidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
6-[2-oxo-2-(piperidin-1-yl)ethyl]-5,6-dihydro-1,6-naphthyridin-5-one
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}urea
6-{4-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
2-[5-(furan-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(2S,3S)-2-{[1-(4-fluorophenyl)propan-2-yl]amino}-3-methylpentan-1-ol
(1S,5R)-3-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
benzyl 3-(oxane-4-amido)pyrrolidine-1-carboxylate
N-[2-(2,4-difluorophenyl)-1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-oxazole-4-carboxamide
4-cyclobutyl-N-[3-(1H-imidazol-1-yl)butyl]-6-methylpyrimidin-2-amine