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propan-2-yl 2-chloro-5-[(2S)-oxolane-2-amido]benzoate
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
6-(3-hydroxyazetidin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
(2R,6S)-4-(2-ethylpyrimidine-5-carbonyl)-2,6-dimethylmorpholine
5-[(5-phenylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(4aR,7aS)-1-methyl-4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidine-1-carboxamide
1-[1-(2-methoxyethyl)piperidine-4-carbonyl]-4-(4-methoxyphenoxy)piperidine
2,2-dimethyl-N-[(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]propanamide
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-[(5-methylthiophen-2-yl)methyl]-1-(pyridin-2-ylmethyl)urea
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(piperidin-1-yl)butanamide
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(furan-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
3-[1-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(2,2-dimethyloxan-4-yl)benzamide
8-(but-3-enoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-phenyl-3-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-(dimethyl-1,2-oxazol-4-yl)-5-{1-[(2E)-hex-2-en-1-yl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-[4-(2-methylpropyl)piperazin-1-yl]-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-(1,4-dioxane-2-carbonyl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-(propan-2-yl)-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-1H-pyrazole-3-carboxamide
({3-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
4-{2-[2-(quinolin-8-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-chlorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-[1-(2-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
ethyl 4-[(4-methoxyphenyl)methyl]-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxylate
3-{2-oxo-2-[4-(2-phenylethyl)piperidin-1-yl]ethyl}-4-(pyridin-2-ylmethyl)piperazin-2-one
3-(2-ethyl-1H-imidazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
4-{1-[(8-methoxy-2H-chromen-3-yl)methyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
(4aS,8aR)-6-[(2-chloro-6-methylphenyl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
8-cyclopropanecarbonyl-2-(5-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-cyclopropyl-1-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
2-ethyl-9-[(1-methyl-1H-indol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 1-benzyl-5-[(1-hydroxypropan-2-yl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 5-[({5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazol-3-yl}formamido)methyl]furan-2-carboxylate
4-chloro-N-(2-methoxyethyl)-1-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-cyclobutaneamido-N-[(1-cyclopentylpiperidin-4-yl)methyl]benzamide
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methoxypropanamide
3-[3-(trifluoromethyl)phenyl]-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
2-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[4-(hydroxydiphenylmethyl)piperidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(oxolan-2-ylmethyl)propylamine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-(methylsulfanyl)benzamide
1-(cyclopropylmethyl)-5-(3-methylfuran-2-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(adamantan-1-yl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]acetamide