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2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
2-methyl-7-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-4-oxobutanamide
4-{4-[(5-chloro-2-fluorophenyl)methyl]piperazin-1-yl}butan-1-ol
1-(3-methylpyridin-4-yl)-4-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
4-[(3,5-dimethoxyphenyl)methyl]-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
3-(hydroxymethyl)-1-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]pyrrolidin-3-ol
2-phenyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide
N-[3-(benzylsulfanyl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
1-[3-(piperidin-3-yl)benzoyl]-4-(pyridin-3-yl)piperazine
(2S)-2-{2-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}propanamide
2,2-dimethylpropyl (4aS,7aR)-4-[2-(dimethylamino)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
2-{3-[3-(6-methoxypyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}-N-(pyrazin-2-yl)acetamide
N-[2-(3-fluorophenyl)-2-hydroxyethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
3,5-dichloro-4-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]pyridine
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-{1-[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
2-({4-[6-(azepan-1-yl)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
N-(1-{2-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(2-methoxyphenyl)acetamide
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-methyl-2-phenyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(thiophen-2-yl)propanamide
dimethyl({[(3S,4R)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
3-methoxy-5-[4-(1H-pyrazol-5-yl)phenyl]pyridine
2-{4-[(4-ethynylphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(2-methoxyethyl)-3-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]propanamide
3-{[(3R,4R)-3-hydroxy-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl]methyl}-4H-chromen-4-one
2-(4-chlorophenyl)-4-(3-phenyl-1H-pyrazole-5-carbonyl)morpholine
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)oxane-2-carboxamide
1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-2-(pyridin-4-yl)ethan-1-one
N-(1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}cyclopentyl)aniline
2-methyl-3-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}phenol
5-{1-[3-(4-methoxyphenyl)propanoyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
N-cyclopentyl-6-(methoxymethyl)-N-[(2-methoxyphenyl)methyl]pyridine-2-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide
1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(naphthalen-2-yl)ethan-1-one
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
2-(4-fluorophenoxy)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
8-methoxy-2-methyl-4-[4-(trifluoromethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(1H-indol-2-ylmethyl)-1-methyl-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1,5-dimethyl-4-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
3-phenyl-1-{1-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}propane-1,2-dione
(1R,5S)-3-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aR,7aS)-4-[4-(hydroxymethyl)benzoyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
5-methyl-1-propyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-4-carboxamide