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3-(2-fluorophenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-{[4-(3-chlorophenyl)-5-({methyl[(2E)-2-methylbut-2-en-1-yl]amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
2-{2-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]phenyl}-1H-imidazole
4-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-(methoxymethyl)-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
1-(2-{methyl[(6-methylpyridin-2-yl)methyl]amino}ethyl)piperidin-2-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}acetamide
4-cyclobutyl-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-6-methylpyrimidin-2-amine
{1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
2-amino-4-(2-methoxypyrimidin-5-yl)-6-methyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(2-fluorophenyl)methyl]-3-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl}propanamide
2-[methyl({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl})amino]ethan-1-ol
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrrol-2-yl)pyridine
2-({2-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
4-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]-1-(propan-2-yl)pyrrolidin-2-one
5-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]-N-(propan-2-yl)pyrimidin-2-amine
1-(furan-2-ylmethyl)-2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazole
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]piperidine-4-carboxamide
3-fluoro-N-[(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
(2S,4S)-4-amino-N-ethyl-1-{[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({2-[4-(trifluoromethyl)phenyl]ethyl})amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-methylphenyl)methyl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
4-(2-methoxyethyl)-1-[(3-methylphenyl)methyl]-1,4-diazepan-5-one
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
1-[(1S,5R)-6-(anthracene-9-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[(3R,5S)-1-cyclohexyl-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[2-(5-methylthiophen-2-yl)ethyl]urea
1-(2-methyl-1,3-thiazole-4-carbonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
5-methoxy-2-({4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-4H-pyran-4-one
methyl 3-(3,4-dimethylbenzoyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-{2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}phenyl)imidazolidin-2-one
ethyl 1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylate
3-amino-1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(naphthalen-2-ylmethyl)pyrrolidin-3-yl]methanol
1-(4-{2-[3-(2-methylphenoxy)azetidin-1-yl]-2-oxoethoxy}phenyl)propan-1-one
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-3-(benzylsulfanyl)propan-1-one
6-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
(1R,5R)-N,N-dimethyl-6-[3-(pyridin-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-(4-{[5-(4-chloro-2-fluorophenyl)furan-2-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-(3-{[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl}phenyl)ethan-1-one
3-cyano-N-[1-(3-methylpyridin-2-yl)ethyl]benzamide
2-methoxy-5-oxo-6-[4-(pyrrolidin-1-yl)butyl]-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-{[8-(4-methylpyrimidin-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}furan-2-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(1,2-benzoxazol-3-yl)acetyl]-1,4-diazepane-6-carboxylic acid
(3-benzyl-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-yl)methanol
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-fluorophenyl)ethan-1-one
1-(cyclobutylmethyl)-3-hydroxy-3-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
3-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
(3aS,6aS)-2-(1-benzofuran-2-ylmethyl)-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,8aR)-6-[(5-ethylpyridin-2-yl)methyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one