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2-benzyl-N-({3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-1,3-thiazole-4-carboxamide
1-{3-[(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)methyl]phenyl}ethan-1-one
N'-cyclopentyl-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]butanediamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(2-methylpyridine-3-carbonyl)piperidin-3-ol
4-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
N-({1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)cyclohexanecarboxamide
4-(furan-2-yl)-2-{4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-5-(propan-2-yl)-1H-pyrazol-1-yl}pyrimidine
1-(2-methoxyphenyl)-4-[3-(2-methylphenyl)propanoyl]piperazin-2-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[(4-methylphenyl)sulfanyl]-1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
N,N-dimethyl-6-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazine-2-carboxamide
N-[2-(oxolane-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-4-(trifluoromethyl)benzamide
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
N-[(6-chloropyridin-3-yl)methyl]-1-[2-(dimethylamino)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
methyl 2-(1-{[3-(2-methoxyacetamido)-2-methylphenyl]carbamoyl}pyrrolidin-3-yl)acetate
N-[3-(azepan-1-yl)propyl]-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
ethyl 4-[4-(4-{[3-(1H-pyrazol-1-yl)propyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
9-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylspiro[2.4]heptane-1-carboxamide
N-(4-{[(1R,5S,6S)-6-(4-methylpiperazine-1-carbonyl)-3-azabicyclo[3.1.0]hexan-3-yl]methyl}phenyl)acetamide
1-(2,2-dimethylpropyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
(3aS,6aR)-5-[(2,4-difluorophenyl)methyl]-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)oxane-4-carboxamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N,N-dimethyl-1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-amine
N-cyclobutyl-3-({3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}sulfonyl)benzamide
2-(cyclohex-1-en-1-yl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
4-({1-[3-(4-methylphenyl)phenyl]piperidin-4-yl}amino)butan-1-ol
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)[2-(oxan-4-yl)ethyl]amine
5-acetyl-3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
5-cyclopropyl-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
2-[2-(piperidin-1-ylmethyl)phenoxy]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-methyl-N-(1-methylpyrrolidin-3-yl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
6-ethyl-2-methyl-4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}quinoline
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
4-methyl-2-oxo-5-[3-(2-phenylacetyl)piperidine-1-carbonyl]-1,2-dihydropyridine-3-carbonitrile
(3aR,6aR)-N-[(1-ethyl-1H-indazol-3-yl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(aminomethyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
N3-methyl-N5-[(4-methylphenyl)methyl]-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
4-{4-[(2-cyclohexylpyrimidin-5-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
3-(cyclopropylmethyl)-1-(4-ethylphenyl)-3-(2-methoxyethyl)urea
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-fluorophenyl)piperazine
ethyl 4-[2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetyl]piperazine-1-carboxylate
5-ethyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
8-fluoro-N-[(3-hydroxy-4-methoxyphenyl)methyl]-N-methylquinoline-2-carboxamide
2-{4-[3-cyclopropyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenoxy}acetamide