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N-[(5-methylpyrazin-2-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
{1-[1-(3-fluoro-4-methylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanamine
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1-(pyridin-2-ylmethyl)piperidin-2-one
4-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
5-(5-acetylthiophene-2-carbonyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-2,3-dihydro-1H-inden-2-amine
(3S,4R)-4-(3-fluorophenyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}pyrrolidine-3-carboxylic acid
methyl (2R,4S)-1-[(4-ethylphenyl)methyl]-4-hydroxypiperidine-2-carboxylate
[(2-ethoxypyridin-3-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-(1-methoxybutan-2-yl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-ethoxy-3-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
7-methyl-2-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
(3aS,6aS)-2-(1H-imidazole-2-carbonyl)-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-methoxy-N-({1-[3-(1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
ethyl 4-{[2-(2-chloro-6-methylphenoxy)ethyl]amino}piperidine-1-carboxylate
1-ethyl-3-(piperidine-1-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(2S)-1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidine-2-carbonyl]morpholine
N-[(2R,3R)-1'-(2,5-dimethylbenzoyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
3-methyl-3-[2-(oxan-2-yl)ethyl]-1-phenylurea
5-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
4,4,4-trifluoro-1-[4-(4-methoxyphenoxy)piperidin-1-yl]butan-1-one
2-[(3-chlorophenyl)methyl]-N-(6-hydroxy-6-methylheptan-2-yl)-1,3-benzoxazole-6-carboxamide
2-(5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-pyrazol-3-yl)phenol
methyl 3-ethyl-2-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-3H-imidazo[4,5-b]pyridine-6-carboxylate
2-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(4aS,8aS)-2-[4-(2-fluorophenyl)benzoyl]-decahydro-2,7-naphthyridin-4a-ol
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-6-(propan-2-yl)pyridazin-3-amine
3-(diphenylmethyl)-5-(furan-3-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-(2-acetamidoethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
4-methyl-N-{3-[3-(3-methylphenoxy)azetidin-1-yl]-3-oxopropyl}benzamide
1-ethyl-4-[3-(4-fluorophenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
2-(3-chloro-4-hydroxyphenyl)-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-methylpiperidine
2-ethoxy-3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}pyridine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-[1-(3-methylphenyl)piperidin-4-yl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
2-[1-(propan-2-yl)piperidin-4-yl]-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
4-[4-(3-chlorophenyl)-3-oxopiperazine-1-carbonyl]oxane-4-carbonitrile
N-[(3R,4R)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
5-fluoro-1,3-dimethyl-N-[4-(methylamino)butyl]-1H-indole-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-ethoxypropanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-(4-{[1-(3-methylpyridin-2-yl)propan-2-yl]amino}piperidin-1-yl)pyridine-3-carbonitrile
3-{[(3S,4R)-3-cyclopropyl-4-acetamidopyrrolidin-1-yl]sulfonyl}benzoic acid
methyl 5-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]methyl}acetamide
1-(1-benzylpiperidin-4-yl)-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
(4-{[(4-cyclobutyl-6-methylpyrimidin-2-yl)(methyl)amino]methyl}oxan-4-yl)methanol
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-3-yl]propanoate