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2-(1-methyl-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-cyclopentyl-1-[3-(3-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine
1-[(3-fluorophenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
(2S,4R)-1-[(2,6-difluorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl N-(1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl)carbamate
N-[(2R,3R)-2-methoxy-1'-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
2-(1-{[(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-6-fluorobenzamide
N-ethyl-2-[1-(2-methylbutyl)-3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl]propanamide
3-[5-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-[3-chloro-2-(propan-2-yloxy)phenyl]-1-[2-(pyrazin-2-yl)ethyl]urea
6-oxo-N-[1-(pyridin-4-yl)propyl]-1,6-dihydropyridine-3-carboxamide
1-{[3-(pyridin-2-yl)phenyl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
3-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5,8-dimethyl-2-({[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]amino}methyl)quinolin-4-ol
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1-ethylpiperidine-2-carboxamide
3-methyl-7-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(2-chloro-3-methoxyphenyl)-1-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)urea
1-[2-(3-ethoxyphenoxy)ethyl]-4-(oxolan-2-ylmethyl)piperazine
4-chloro-N-methyl-2-propanamido-N-propylbenzamide
4,6-dimethyl-1-{2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
N-[2-(2,4-difluorophenyl)-1-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
methyl 4-{[(4aR,8aS)-1-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-6-yl]methyl}benzoate
7-(1,3-benzothiazol-2-yl)-4-(3-fluoropropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2,6,8-trimethyl-4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]quinoline
7-(2-methylphenyl)-4-(quinoxalin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[(5-chlorothiophen-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
(1S,5R)-3-methyl-6-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3,6-diazabicyclo[3.2.2]nonane
3-(4-hydroxyphenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-pyrazole-5-carboxamide
4-{4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine-1-carbonyl}morpholine
2-(4-hydroxypiperidin-1-yl)-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
[3-({1-[2-(1H-imidazol-2-yl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-cyclopropyl-3-{ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]sulfamoyl}benzamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-2-carbonyl)pyrrolidin-3-yl]-4-methylpyrimidine-5-carboxamide
({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-chloro-N-(1-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
3-(3,4-difluorophenyl)-5-(morpholine-4-sulfonyl)benzoic acid
1-[2-(4-methoxybenzenesulfonamido)ethyl]-N-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
2-[3-(dimethylamino)propyl]-9-[6-(dimethylamino)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-({1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)-2-methylpropanamide
{[4-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)phenyl]methyl}dimethylamine
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)propanamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
3-(2-ethylphenoxy)-1-(thiophene-2-carbonyl)azetidine
5-(2,6-dimethylphenoxymethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-1,2-oxazole-3-carboxamide