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2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(1,3,5-triazin-2-yl)piperazin-1-yl]ethan-1-one
2-(3-methoxyphenyl)-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
4-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
3-[1-(1-methylpiperidin-4-yl)-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-3-yl]pyridine
(2R,4S)-1-(3,5-dimethylbenzoyl)-4-hydroxypiperidine-2-carboxylic acid
N-(furan-2-ylmethyl)-N-methyl-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{[2-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-4-(piperidin-3-yl)benzamide
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-4-methyl-N-(pyridin-4-ylmethyl)benzamide
(3S,4S)-3-hydroxy-4-[4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
2-(azocane-1-carbonyl)-6-(2,5-dimethylfuran-3-yl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
3-[2-(4-fluorophenoxy)ethyl]-N-methylbenzamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
7-cyclohexyl-2-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-cyclopentyl-5-oxo-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}pyrrolidine-3-carboxamide
2-chloro-N-ethyl-5-[({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}carbamoyl)amino]benzamide
9-(2,6-dimethoxypyrimidine-4-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-(1-hydroxy-2-methylpropan-2-yl)-1,3-oxazole-4-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]propanamide
8-[3-(2-fluorophenyl)-3-phenylpropanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{2-[methyl({5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl})amino]ethyl}cyclopentan-1-ol
(4S)-1-cyclobutanecarbonyl-3,3,4-trimethylpiperidin-4-ol
1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2,6-dimethyl-4-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}quinoline
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylcyclohexane-1-carboxamide
3-chloro-2-{[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]methyl}-1H-indole
5-ethyl-N-[1-(1,3-thiazol-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
6-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(3-methoxypropanoyl)-N-(oxolan-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[3-(furan-2-yl)phenyl]-1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidine-4-carboxamide
2-(3-fluorophenoxymethyl)-8-(1-methyl-1H-pyrazole-5-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
4-[({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]-2-methoxypyridine-3-carbonitrile
N-(2-{1-ethyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-4-fluorobenzamide
6-[2-(cyclohex-1-en-1-yl)acetyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(1R,5R)-3-(1-benzofuran-5-carbonyl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane
5-(1-benzyl-1H-pyrazol-3-yl)-N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-methyl-1,3-thiazol-2-amine
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl}){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
2-[1-cyclopentyl-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
3-{[2-(dimethylamino)ethyl](ethyl)amino}-N-(2-fluorophenyl)propanamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(1-methylpiperidin-2-yl)acetamide
3-(1-methyl-1H-imidazol-2-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
benzyl N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)-5-{1-[2-(thiophen-2-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N,6-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine