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N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-3-fluoro-N-(oxolan-2-ylmethyl)benzamide
3-{[2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}acetamide
4-{2-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidine-1-carbonyl]phenyl}morpholine
ethyl 4-benzylpiperidine-4-carboxylate
5-[benzyl(methyl)amino]-2-(2,3-dihydroxypropyl)-2,3-dihydropyridazin-3-one
3-[(2,1,3-benzothiadiazol-5-ylmethyl)amino]-N-(4-methoxyphenyl)-5-(methylsulfamoyl)benzamide
N-{2-[(2,3-dimethylquinoxalin-6-yl)formamido]ethyl}pyridine-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
N-(1-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
1-(1,4-dioxan-2-ylmethyl)-4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazole
N-[2-(2,4-difluorophenyl)-1-{1-[(2,5-difluorophenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
2-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-4-(1H-pyrrol-1-yl)phenol
3-tert-butyl-4-(1H-imidazol-2-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
8-(6-methylpyridine-2-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-fluoro-N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-{1-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]piperidin-3-yl}benzoic acid
3-[1-(2-chlorobenzoyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
N-(3-hydroxy-3-phenylpropyl)-N,2,5-trimethyl-1,3-thiazole-4-carboxamide
methyl 2-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetate
2-phenyl-N-(piperidin-4-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
1-(4-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2,6-difluorobenzamide
N,3,5-trimethyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]adamantane-1-carboxamide
(3S,4R)-4-methyl-1-[3-(morpholin-4-yl)benzoyl]piperidine-3,4-diol
N-(2-methyl-1-{7-[2-(phenylsulfanyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
2-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-cyclobutanecarbonyl-N-[2-(1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[3-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)propyl]phenol
4-{3-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3-oxopropyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[2-methyl-6-(propan-2-yl)phenyl]-2-{[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]amino}acetamide
2-[2-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
8-[(2-fluoro-4-methoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{2-[5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
N-({1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidin-3-yl}methyl)acetamide
2-[2-({[5-(methylcarbamoyl)furan-2-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
5-ethyl-5-[1-(quinoxaline-5-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-cyclopropyl-5-{1-[3-(pyrazin-2-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-methyl-4-phenyl-3-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-[(cyclobutylformamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
2-(5-oxopyrrolidin-2-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
N-methyl-N-{1-[1-(3-methylbenzoyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-2-(1H-pyrazol-1-yl)acetamide
N-cyclobutyl-1-(3-phenylphenyl)piperidin-4-amine
3-{1-[(2-hydroxy-3-methylphenyl)methyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2,3-dimethylquinoxaline-6-carbonyl)-4-(4-fluorophenyl)piperidin-4-ol