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3-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}-6-methyl-4H-chromen-4-one
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)but-3-enamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-4-(trifluoromethyl)benzamide
[2,4,6-trimethyl-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)phenyl]methyl acetate
4-{5-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
5-benzyl-5-{3-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-(cyclohexylmethyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
2-methoxy-N-methyl-5-({[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}amino)benzamide
N-(furan-2-ylmethyl)-2-(methoxymethyl)-N,1-dimethyl-5-(2-phenylacetamido)-1H-1,3-benzodiazole-7-carboxamide
6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N,N-dimethylpyrimidin-4-amine
N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)pyrazine-2-carboxamide
1-(4-benzylpiperazin-1-yl)-3-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}propan-1-one
7-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(3aR,6aR)-2-(2-methoxyacetyl)-N-methyl-N-(pyrazin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(4S)-3,3,4-trimethyl-1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]piperidin-4-ol
1-(1-methylpiperidin-4-yl)-N-(1H-1,2,4-triazol-3-ylmethyl)piperidine-3-carboxamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
1-(4-fluorophenyl)-4-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
N-[(1R,2R)-2-hydroxycyclohexyl]-N-propyl-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
(1S,5R)-3-(furan-3-ylmethyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{3-cyclopropyl-5-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-1,2,4-triazol-1-yl}-6-methylpyridine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2,4-dimethylbenzene-1-sulfonamide
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]urea
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-[2-(5-methylfuran-2-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(4aS,7aR)-4-(furan-2-carbonyl)-6,6-dioxo-N-(propan-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-[2-(1H-imidazol-1-yl)propyl]-1-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
4-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-[2-(dimethylamino)ethyl]pyrrolidin-2-one
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[5-(oxan-2-yl)thiophen-2-yl]methyl}amine
ethyl 3-[(4-fluorophenyl)methyl]-1-(4-methoxy-4-oxobutanoyl)piperidine-3-carboxylate
1-(2-cyclohexylethyl)-3-hydroxy-3-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)piperidin-2-one
(1R,5R)-6-benzyl-N-(2-methoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(oxolan-2-ylmethoxy)ethan-1-one
5-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-2-methoxypyridine
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(4-methylpiperazin-1-yl)propanamide
methyl 5-(2-chloropyridine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-(dimethylamino)-1-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]-2-(4-methylphenyl)ethan-1-one
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-(2-phenylethyl)piperidine-1-carboxamide
2-(2-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
2-(morpholin-4-yl)-1-{4-[4-(1H-pyrazol-5-yl)phenyl]phenyl}ethan-1-ol
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(3-methoxypiperidin-1-yl)pyridine
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-[(5-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(dimethylamino)ethyl]-N-[(4-methylpyridin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-[5-methoxy-2-({[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-(2,3-dihydro-1H-inden-2-yl)-5-[(2-methoxyethoxy)methyl]-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazole
N-(2-hydroxyethyl)-3,4,7-trimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-indole-2-carboxamide
8-[(6-chloroquinolin-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-benzyl-5-[(3-hydroxy-4-methoxyphenyl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(4-methyl-1H-pyrazol-3-yl)-N-{2-[2-(methylcarbamoyl)ethyl]phenyl}piperidine-1-carboxamide