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(1S,5R)-N-methyl-7-oxo-N-phenyl-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[1-(naphthalen-1-yl)ethyl]propanamide
N-({7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
(1S,5R)-1,3,3-trimethyl-6-(4-methylpyrimidine-5-carbonyl)-6-azabicyclo[3.2.1]octane
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
1-{4-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-4-oxobutyl}piperidin-2-one
3-(1-ethyl-2-methyl-1H-indol-5-yl)-1-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
1-(3-methylbutyl)-8-{[4-(methylsulfanyl)phenyl]methyl}-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-(naphthalen-2-yl)acetamide
N-(furan-2-ylmethyl)-N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
2-{4-[4-(1-methoxyethyl)phenyl]phenyl}-5-methyl-1,3,4-oxadiazole
methyl 2-(diethylsulfamoyl)-6-(quinolin-5-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3,4-difluorobenzamide
(2E)-N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylbut-2-enamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-methyl-3-phenylbutanamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(methylamino)pyridine-4-carboxamide
3-methyl-7-(5-propyl-1,2-oxazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
6-{[ethyl(oxan-4-yl)amino]methyl}pyridine-2-carboxylic acid
1-cycloheptyl-6-oxo-N-[2-(propan-2-yloxy)ethyl]piperidine-3-carboxamide
1-(1'-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-{1-[1-(2,5-dimethylbenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(5-methyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(3-methylthiophene-2-carbonyl)piperidine-2-carboxamide
ethyl 1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-2-carboxylate
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(furan-2-yl)propanamide
3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one
N-(cyclopropylmethyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-(1-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
2,3-difluoro-5-(1H-indazol-1-yl)phenol
4-[({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1-(propan-2-yl)pyrrolidin-2-one
ethyl 5-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
N,N-diethyl-1-{[4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-3-carboxamide
3-[(3,4-dimethylphenyl)methyl]-9-methoxy-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(naphthalen-2-ylmethyl)piperidine
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(pyrrolidine-1-carbonyl)pyridine
6-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(propan-2-yl)-4-({[4-(propan-2-yl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-{[(3-chloro-4-methylphenyl)carbamoyl]amino}-N-methylcyclohexane-1-carboxamide
N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
7-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,3-diazepane-2,4-dione
2-{4-[(6-chloro-2H-chromen-3-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
3-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1-[4-(methylsulfanyl)phenyl]urea
1-(2-methanesulfonylethyl)-4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperazine