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5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-1H-pyrazole-4-carboxamide
2-(pyridin-4-yl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-(2-methylpropyl)-1,2,4-oxadiazole
1-[(2-ethoxyphenyl)methyl]-3-(pyrrolidin-1-yl)pyrrolidine
(4aS,8aR)-1-(3-hydroxypropyl)-6-(3-methylbut-2-enoyl)-decahydro-1,6-naphthyridin-2-one
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
4-[(3-fluorophenyl)methyl]-3-{2-[4-(3-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
2-{1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
[(1-benzylpiperidin-4-yl)methyl]({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-2,6-dimethylphenyl acetate
5-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1-methyl-1H-1,2,3-benzotriazole
8-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-3-[2-(dimethylamino)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{4-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
1-[5-(2,3,4-trimethoxyphenyl)furan-2-carbonyl]piperidine
N-[1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
9-[(3-chlorophenyl)methyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
6-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-2-oxo-N-[1-(thiophen-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
7-(1,3-benzothiazol-2-yl)-9-methoxy-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-ethoxy-5-[(4-methylphenyl)methyl]-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-ethyl-4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
5-{2-azaspiro[4.4]nonan-2-ylmethyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
1-(2-{4-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
methyl 3-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
[(2S,6S)-4-(5-methoxyfuran-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-fluoro-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-sulfamoylbenzamide
4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
7-[1-(benzenesulfonyl)cyclopropanecarbonyl]-3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
3,4,7-trimethyl-2-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1H-indole
N-benzyl-N-butyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxylic acid
2-cyclohexyl-5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}pyrimidine
2-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-benzyl-N-(2-hydroxyethyl)propanamide
(1R,3S)-3-(2-hydroxyethoxy)-7-(3-methyl-1-benzothiophene-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-[2-(4-chlorophenyl)ethyl]-N-(1H-imidazol-2-ylmethyl)-6-oxopiperidine-3-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propan-1-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxy-2-methylbenzamide
2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]-2-[3-(methylsulfanyl)phenyl]acetic acid
5-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)furan-2-carboxamide
3-(piperazine-1-carbonyl)-N-[2-(pyridin-4-yl)ethyl]benzene-1-sulfonamide
5-(4-methyl-1,4-diazepan-1-yl)-2-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,3-dihydropyridazin-3-one
4-methoxy-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
6-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-{1-[(1-phenyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}benzoic acid
N-[3-(4-methoxyphenyl)propyl]-6-(morpholin-4-yl)pyridine-3-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2,4-difluorobenzene-1-sulfonamide
(4aR,8aS)-1-(2,2-diphenylethyl)-6-(furan-2-carbonyl)-decahydro-1,6-naphthyridin-2-one