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5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-[3-(propan-2-yloxy)propyl]pyrrolidin-2-one
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-2-ethoxypyridine
5-methyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-(4-methylpent-3-en-1-yl)piperidin-2-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-methyl-N-(propan-2-yl)piperidine-3-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]propan-1-one
6-[5-chloro-2-(propan-2-yloxy)phenyl]-N,N-dimethylpyridine-3-carboxamide
1-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,3-thiazole
1-[3-(cyclopentyloxy)phenyl]-3-methyl-3-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-(1-{4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
[4-({1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-(quinoxalin-6-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-(cycloheptylamino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(piperidin-1-yl)-2-[4-(quinolin-2-ylmethyl)piperazin-1-yl]ethan-1-one
N,1-dimethyl-5-{methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-benzyl-1-(cyclopropylmethyl)-3-ethyl-1,4-diazepan-5-one
2-(1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazol-4-yl}-N-methylformamido)-N,2-dimethylpropanamide
N-[(2R,3R)-1'-{[3-(2-hydroxyethoxy)phenyl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
2-(4-{[(2,6-dimethylmorpholin-4-yl)sulfonyl]amino}-3,5-dimethyl-1H-pyrazol-1-yl)acetic acid
2,4-dimethyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1,3-thiazole-5-carboxamide
N-{[3-(methylsulfanyl)phenyl]methyl}-4-sulfamoylbenzamide
3-{4-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]phenyl}-1,3-oxazolidin-2-one
5-(methoxymethyl)-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
2-(2,6-dimethoxy-4-methylphenyl)-2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetic acid
3-(4-chlorophenyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]-3-phenylpropanamide
2-(dimethylamino)-1-[4-(2-methanesulfonylethyl)piperazin-1-yl]-2-(2-methylphenyl)ethan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-methoxyacetamide
4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(5-methylfuran-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(adamantan-1-yl)-N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole-3-carboxamide
3-[2-(1-benzylpyrrolidin-3-yl)ethyl]-1-(3-methoxyphenyl)urea
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-(4-methanesulfonylpiperazine-1-carbonyl)-5,6-dimethyl-1,2-dihydropyridin-2-one
2-({[3-(dimethylamino)thiolan-3-yl]methyl}amino)-N-(pyrazin-2-yl)acetamide
2-[1-methyl-3-(pyridin-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
4-(1-benzofuran-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-{3-[methyl(phenyl)amino]propyl}-2-(trifluoromethyl)pyrimidin-4-amine
1-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
methyl 4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(1-phenylcyclopropyl)propanamide
2-{4-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
ethyl 2-({1-[4-({[2-(3-fluorophenyl)ethyl]carbamoyl}methyl)phenyl]piperidin-4-yl}(methyl)amino)acetate
1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
1-(4-{[4-(5-fluoro-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
1-[4-(morpholin-4-yl)-3-(1H-pyrazol-3-yl)phenyl]ethan-1-one