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(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)acetyl]pyrrolidine-3-carboxylic acid
3-[5-(dimethyl-1,2-oxazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-3-(1-methylpiperidin-2-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-butyl-3-{[(3S)-3-acetamidopyrrolidin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
2-(2-methoxyphenoxy)-2-methyl-1-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}propan-1-one
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
4-[(4-methoxynaphthalen-1-yl)methyl]-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
2-(4-methylphenyl)-5-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrimidin-4-ol
2-methoxy-1-[1'-(1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-{3-[4-(5,6-dimethylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]quinoline
N-(1-benzothiophen-5-ylmethyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-{2-[(cyclohex-1-en-1-ylmethyl)amino]propyl}-3,4-dihydroquinazolin-4-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide
2-{[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]sulfonyl}benzonitrile
1-tert-butyl-4-[({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)methyl]pyrrolidin-2-one
7-{[5-(methoxymethyl)furan-2-yl]methyl}-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(1S,6R)-3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3,9-diazabicyclo[4.2.1]nonane
N-[(2,3-dimethoxyphenyl)methyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-[(4-methyl-1H-imidazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
4-[(3R,5R)-5-[4-(pyridin-3-yl)piperazine-1-carbonyl]piperidine-3-carbonyl]morpholine
N-[4-(4-{[1-(thiophen-2-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
4-[(4-methanesulfonylphenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
2-{3-[2-(4-ethoxyphenyl)pyridin-4-yl]pyrrolidin-1-yl}acetic acid
2-[(3S,4R)-3-cyclopropyl-4-{[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}pyrrolidin-1-yl]acetamide
(5S,9aS,9bS)-5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-chloro-4-{[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]methyl}phenol
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
1-{1-[(2E)-3-(5-chloro-2-hydroxyphenyl)-2-methylprop-2-en-1-yl]piperidin-3-yl}pyrrolidin-2-one
(1S,5R)-6-benzyl-3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,4-oxazepan-6-ol
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2-methyl-1-(propan-2-yl)piperazine
N-{2-[({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}pyridine-3-carboxamide
N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-butyl-4-(cyclopropylamino)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
(4aS,7aR)-1-(2-cyclohexylacetyl)-4-[2-(dimethylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl (2S,4R)-4-hydroxy-1-[3-(2-methyl-1H-indol-1-yl)propanoyl]pyrrolidine-2-carboxylate
N-(4-methoxyphenyl)-2-{4-[(2E)-3-phenylprop-2-en-1-yl]morpholin-3-yl}acetamide
N-({1-[(2E)-4-methylpent-2-enoyl]piperidin-3-yl}methyl)furan-2-carboxamide
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(2,5-dimethoxyphenyl)acetamide
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-cyclopropylpropanamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(1H-indole-2-carbonyl)-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(cyclopropanesulfonyl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-ethyl-N-[3-(morpholin-4-yl)propyl]propanamide
1-[(2-ethoxyphenyl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]benzonitrile