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1-(5-ethyl-2-methylpyrimidin-4-yl)-4-(furan-3-carbonyl)-1,4-diazepane
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,2-dihydroquinolin-2-one
2-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-4-methoxyphenol
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
4-(benzyloxy)-1-[2-(pyrrolidin-1-yl)benzoyl]piperidine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-{[5-(2-chlorophenyl)-4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4,5-dimethyl-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyrimidine
methyl 4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine-1-carboxylate
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(pyridin-3-ylmethyl)pyridin-2-amine
3-(2-chlorophenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-phenylpropanamide
6-fluoro-2-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)quinoline
7-(3-chlorophenyl)-4-[(4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(carbamoylmethyl)phenyl]-4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carboxamide
(1R)-2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-phenylethan-1-ol
2-methoxy-4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]phenol
1-(2-ethoxyethyl)-5-[4-(2-methoxyethyl)piperidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(3-benzoylpiperidin-1-yl)-5-(1H-imidazol-1-ylmethyl)pyridine
N-[2-(3-methoxyphenyl)ethyl]-6-(quinolin-6-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidine-3-carboxylate
1-tert-butyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinolin-2-one
N-(2-methylprop-2-en-1-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
7-(2-methylphenyl)-4-(5-methylthiophene-2-carbonyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1,3-oxazole-4-carboxamide
4-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-ethyl-3-(1H-indol-3-yl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
1-(3-fluorophenyl)-4-(1H-imidazol-2-yl)-3-(5-methylfuran-2-yl)-1H-pyrazole
4-fluoro-3-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
2-[2-(dimethylamino)ethyl]-8-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane-6-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
ethyl 4-(3-{[(3-{2-azabicyclo[2.2.1]hept-5-en-2-yl}propyl)amino]methyl}-6-methylquinolin-2-yl)piperazine-1-carboxylate
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-amine
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-ethyl-3-(propan-2-yl)-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-5-carboxamide
(1S,5R)-6-phenylmethanesulfonyl-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-indole-3-carboxamide
2-[(4-fluorophenyl)methyl]-4-[(4-methoxyphenyl)methyl]morpholine
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[2-(methylsulfamoyl)phenyl]urea
N-cyclobutyl-5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N,N-diethyl-1-{2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}pyrrolidin-3-amine
1-[7-(3-chlorophenyl)-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
(3S,4R)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
(3S,5S,9R)-5-({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}amino)-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
8-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
[5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)furan-2-yl]methanol