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N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[(1R,5S,6S)-3-[(2,6-dimethylmorpholin-4-yl)sulfonyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-(prop-2-en-1-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine-3-carboxylic acid
3-(morpholin-4-yl)-N-[4-(trifluoromethyl)phenyl]piperidine-1-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-[3-(benzyloxy)piperidin-1-yl]propan-1-one
(2S,4S)-1-benzyl-N-ethyl-4-{[(4-methoxy-3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
3-{2-[(4aS,8aS)-decahydroisoquinolin-2-yl]-2-oxoethyl}-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3R,4R)-3-hydroxy-1-(4,4,4-trifluorobutanoyl)piperidin-4-yl]pyridine-4-carboxamide
6-{[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
(3S,5S)-1-[(3-hydroxyphenyl)methyl]-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
5-{4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
2-{5-[(4-methoxy-2,3,6-trimethylphenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-[4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-3,5-dimethyl-1H-pyrazol-1-yl]ethan-1-ol
9-(2-ethoxypropanoyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-1-(2-methoxyethyl)-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
(2S)-2-[(5-methoxy-1-methyl-1H-indol-2-yl)formamido]-2-phenylacetamide
3-({[(3-chlorophenyl)methyl]amino}methyl)-N,N-diethylpyridin-2-amine
(1S,5R)-6-(cyclopropylmethyl)-3-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]acetamide
1-methyl-N-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-2-carboxamide
3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-4-cyclopentylpiperazin-2-one
N-[2-(1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]acetamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
2-phenoxy-N-[4-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
2-methoxy-N,N-dimethyl-5-{[({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)carbamoyl]amino}benzamide
3,6-dimethyl-N-(thiophen-3-ylmethyl)-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-chloro-N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-(pent-4-enoyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-amino-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}pyridine-4-carboxamide
8-{1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1H-imidazol-2-yl}quinoline
(5S,9aS,9bS)-2-cyclopentyl-5-(3,4-dimethylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
2-acetamido-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidine
2-[1-(3-phenylpropyl)-4-(pyrimidin-2-yl)piperazin-2-yl]ethan-1-ol
5-(benzylamino)-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]pyridine
2-[5-(4-phenylpiperidine-1-carbonyl)-1H-pyrazol-3-yl]phenol
2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-methyl-N-[2-(oxan-2-yl)ethyl]benzamide
(1R,4R)-2-{2-[1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-2-azabicyclo[2.2.1]heptane
methyl (2S)-2-{[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)azepan-4-yl]amino}-2-phenylacetate
5-{3-[(2,4-difluorophenyl)methyl]-3-(ethoxycarbonyl)piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
3-hydroxy-3-({[2-(4-hydroxyphenyl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
5-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole