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4-[2-(2-methoxyphenoxy)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-(2-{1-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]piperidin-4-yl}ethyl)acetamide
4-benzyl-3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]piperazin-2-one
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-(naphthalen-1-ylmethyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1,2,4-oxadiazole-5-carboxamide
1-(2-oxo-2-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}ethyl)piperidin-2-one
3-(3-fluorophenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-(3-methylphenyl)-1H-pyrazole
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(3,4-difluorophenyl)propan-1-one
3-(3-methylbut-2-en-1-yl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylic acid
4,6-dimethyl-2-{[2-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]methyl}pyrimidine
5-methyl-1-[4-(4-{[3-(pyridin-2-yl)propyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
[1-(methylsulfanyl)propan-2-yl]({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
5-[(4aS,7aR)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
N-[2-(1H-indol-3-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
N-[1-(ethylcarbamoyl)piperidin-4-yl]-2-(propan-2-yl)pyrimidine-4-carboxamide
5-(4-ethylphenyl)pyrimidin-2-ol
3-({3-[(dimethylamino)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)benzonitrile
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(1,2-oxazol-3-ylmethyl)piperidine-3-carboxamide
3-{2-oxo-2-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethyl}-1,3-thiazolidine-2,4-dione
ethyl 1-{5,8-dimethoxy-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]quinolin-2-yl}piperidine-4-carboxylate
1-(cyclopropylmethyl)-N-(pyridin-2-ylmethyl)-5-{spiro[2.5]octane-1-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(1-{1-[4-(propylamino)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
6-ethyl-2-(morpholin-4-yl)-N-(3,3,3-trifluoropropyl)pyrimidin-4-amine
(1S,5R)-3-(3-methoxypyrazin-2-yl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(4-ethylphenyl)methyl]-N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
5-[3-(furan-2-yl)-3-phenylpropanoyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(dicyclopropylmethyl)({[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-methoxy-N-{1-[1-(4-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-1,2,5-thiadiazole-3-carboxamide
1-{[({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)amino]methyl}cyclohexan-1-ol
N-{[5-(3-chlorophenyl)furan-2-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)methanesulfonamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}propanamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-methyl-N-[2-(piperidin-1-yl)ethyl]-1,2-oxazole-5-carboxamide
2-(1-methyl-1H-pyrrole-2-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
methyl 3-(4-methylpentanoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-cyclopentyl-N-[4-(furan-2-yl)butan-2-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
3-[4-(3-cyanophenyl)-1H-1,2,3-triazol-1-yl]-N-(2,5-dimethylphenyl)propanamide
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
1-(4-hydroxy-1,2-oxazolidin-2-yl)-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-thiazole-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(2-methoxyethyl)-N-methyl-6-oxopiperidine-3-carboxamide
6-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)pyridine-2-carboxylic acid
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-4-(pyridin-2-yl)pyrimidin-2-amine
1-(cyclopropylmethyl)-3-hydroxy-3-[({[4-(morpholin-4-yl)phenyl]methyl}amino)methyl]piperidin-2-one