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2-{5-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
1-(4-benzylpiperazin-1-yl)-3-(1-propylpiperidin-3-yl)propan-1-one
2-{4-[7-chloro-4-(3-methylpiperidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]quinoline
6-(2-hydroxyethyl)-N-(pentan-3-yl)-N-(2-phenylethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-(3-chloro-2-methylphenyl)-5-(5-methoxypentyl)-1H-1,2,4-triazole
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
(2S)-2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]-2-phenylacetamide
N-benzyl-5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]furan-2-carboxamide
N-{[7-fluoro-5-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
N-[(2-chlorophenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-[3-(3-chlorophenyl)phenyl]-1-(pyridine-4-carbonyl)piperidine-4-carboxamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-(4-methoxyphenyl)-7-methyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}quinoline
4-[4-(furan-2-yl)benzoyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
(benzylsulfamoyl)({[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl})amine
5-(2-cyclopentylacetamido)-N-[2-(3-fluorophenyl)ethyl]-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
2-{2-[(3,4-dimethylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetic acid
2-(5-carbamoylthiophen-2-yl)-N-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
5-({6,8-dioxo-2,7-diazaspiro[4.4]nonan-2-yl}methyl)-2-methyl-1H-pyrrole-3-carbonitrile
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(2-methoxyphenyl)ethan-1-one
1-[3-(4-phenylbenzoyl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
1-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N-ethyl-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
4-({[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
(5-{1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(2-ethyl-1H-imidazol-1-yl)-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
1-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)urea
4-[3-(3-ethoxyphenyl)phenyl]-4H-1,2,4-triazole
(4aS,8aR)-6-(isoquinoline-5-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
5-chloro-N-methyl-6-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,6-dihydropyridine-3-carboxamide
2-{4-[(4-methoxy-2,5-dimethylphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
5-(3-methyl-1H-pyrazol-5-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
4-[(3,4-dimethoxypyridin-2-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
1-phenyl-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)spiro[2.4]heptane-1-carboxamide
1-[2-({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amino)ethyl]piperidin-3-ol
5-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazole
ethyl 1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[4-(4-{[2-(3-fluorophenyl)ethyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
2-(2-{imidazo[1,2-a]pyridine-2-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-methylcyclopropane-1-carboxamide
1-benzyl-8-{[4-(furan-2-yl)phenyl]methyl}-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-4-(1H-pyrazol-1-yl)butan-1-one
1-(2-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione