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N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-[2-({3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(trifluoromethyl)morpholine
methyl 3-(2-methoxyacetamido)-1-methyl-5-[(4-methylpentan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(2-propoxyphenyl)ethyl]acetamide
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
3,4-dimethoxy-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
N-[(2,6-difluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-[(2-fluorophenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-1H-imidazole-2-carboxamide
2-(4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-propylpyrimidine-5-carboxamide
3-[1-(1H-indole-5-carbonyl)piperidin-3-yl]benzoic acid
2-methyl-4-(1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-6-(pyrrolidin-1-yl)pyrimidine
6-chloro-3-fluoro-N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-2-methoxyethan-1-one
4-phenyl-3-{[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
2-{3-[4-(benzyloxy)piperidine-1-carbonyl]phenoxy}acetamide
(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}azepan-2-yl)methanol
N-[(3,4-difluorophenyl)methyl]-3-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]propanamide
1-(4-{[2-(furan-2-ylmethoxy)phenyl]amino}piperidin-1-yl)ethan-1-one
2-{1-cyclohexyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-methyl-1H-imidazole
2-(2,4-difluorophenyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]acetamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-(2-propyl-1,3-thiazole-4-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-{4-[1-(3-methylpyridine-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
2-methyl-4-oxo-N-[2-(propan-2-yl)phenyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-4-cyclohexylpiperazine
2-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-N-(thiophen-2-ylmethyl)acetamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
3-[4-(trifluoromethyl)benzoyl]piperidine
1-[5-methoxy-2-({methyl[2-(4-methylphenoxy)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
2-[(3-{[(5-fluoro-1H-indol-2-yl)methyl](methyl)carbamoyl}phenyl)amino]acetic acid
2-[1-methyl-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-[2-(1-{[1-(carbamoylmethyl)-2-methyl-1H-indol-3-yl]methyl}piperidin-2-yl)ethyl]acetamide
5-{[4-(1-benzofuran-5-yl)-1H-1,2,3-triazol-1-yl]methyl}thiophene-2-carboxylic acid
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-3-(1H-imidazol-2-yl)benzamide
N-ethyl-2-[3-(furan-2-yl)-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methylacetamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-benzyl-N-ethyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
N-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-N-methyloxan-4-amine
4-[(3-chloro-4-methoxyphenyl)methyl]-1-phenylpiperazin-2-one
2-ethyl-N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
N-[1-(3,4-dimethoxyphenyl)propyl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(trifluoromethyl)benzamide
N-cyclohexyl-N-(prop-2-yn-1-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
[4-(2-phenylethyl)-1-(thiolan-3-yl)piperidin-4-yl]methanol