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6-(methoxymethyl)-N,1-dimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-N-[(1-{[1-(propan-2-yl)piperidin-4-yl]methyl}pyrrolidin-3-yl)methyl]furan-3-carboxamide
1-[2-(1H-pyrazol-1-yl)butanamido]cyclopentane-1-carboxamide
N-[(2,5-dimethoxyphenyl)methyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2,3-dimethyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]quinoxaline-6-carboxamide
3-[(3-{2-[methyl(2-methylpropyl)amino]ethyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)methyl]benzonitrile
N-(furan-2-ylmethyl)-2-hydroxy-4-methoxy-N-(3-methylbutan-2-yl)benzamide
3-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyridine
1-{[3-(2-methylphenyl)phenyl]methyl}-3-(1H-pyrazol-5-yl)piperidine
1-[cyclohexyl(methyl)amino]-3-[2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-{2-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-{4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]morpholin-3-yl}acetic acid
methyl 3-(2-cyclohexylacetyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,4,4-trifluorobutanamide
{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-4-(oxan-2-ylmethyl)piperidin-4-yl}methanol
(3S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-{2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1H-pyrazol-3-one
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-[(2-fluorophenyl)methyl]-1,4-diazepane
6-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino}-N,N-dimethylpyridine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(pyridin-4-yl)propanamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
4-(2-fluorophenoxy)-1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
methyl 5-(cycloheptylamino)-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 5-[(1-methoxypropan-2-yl)amino]-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(furan-2-yl)-5-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}pyrimidine
2-[4-(dimethylamino)phenyl]-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
N-[2-(2-chlorophenyl)ethyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-methyl-1,3-thiazole-4-carboxamide
3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-4-[(4-phenylphenyl)methyl]piperazin-2-one
8-(2,1,3-benzoxadiazol-4-ylmethyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(2H-1,3-benzodioxol-5-yl)-N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
2-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](thiophen-2-ylmethyl)amino}ethan-1-ol
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methoxy-2-phenylacetamide
6-(2-ethoxypyridin-3-yl)-2,4-dimethylpyridine-3-carbonitrile
1-{2-[(cycloheptylamino)methyl]-5-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
2-{1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
ethyl (4aS,8aR)-6-(4-propylpyrimidine-5-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylate
3-methyl-1-(prop-2-en-1-yl)-4-[(3-propylpyrrolidin-1-yl)methyl]-1H-pyrazole
(1S,5R)-3-acetyl-N-(2,5-dimethylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N'-(2-ethoxyphenyl)-N-methyl-N-(1H-pyrazol-5-ylmethyl)propanediamide
4-({3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-9-yl}sulfonyl)piperazine-2-carboxylic acid
2-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-6-methylpyridine-3-carboxamide
3-(2-chlorophenyl)-N-(2-methanesulfonamidoethyl)-3-phenylpropanamide
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methoxyethan-1-one
methyl 3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoate
3-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]urea
5,6-dimethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{[4-(3-chlorophenyl)-5-{[methyl(pyridin-2-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
2-(pyrrolidin-3-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide